نتایج جستجو برای: molecularmodeling

تعداد نتایج: 3  

Aiyoub Parchehbaf Jadid, Leila Javadi Leila Zarefatin

In this study, we present the work on the physicochemical interaction between the anti-cancer alkaloidberberine (BRB) and DNA with the purpose of designing drugs that interact more with DNA. Molecularmodeling on the complex formed between berberine and DNA presented that this complex was undeniablyfully able of participating in the formation of a stable intercalation site. Besides, the molecula...

Journal: :journal of the iranian chemical research 0
aiyoub parchehbaf jadid department of applied chemistry, ardabil branch, islamic azad university, ardabil, iran leila zarefatin department of applied chemistry, ardabil branch, islamic azad university, ardabil, iran leila javadi department of applied chemistry, ardabil branch, islamic azad university, ardabil, iran

in this study, we present the work on the physicochemical interaction between the anti-cancer alkaloidberberine (brb) and dna with the purpose of designing drugs that interact more with dna. molecularmodeling on the complex formed between berberine and dna presented that this complex was undeniablyfully able of participating in the formation of a stable intercalation site. besides, the molecula...

2014
Kellie S. Rath Shan K. Naidu Pushpa Lata Hemant K. Bid Brian K. Rivera Georgia A. McCann Brent J. Tierney Adam C. ElNaggar Veronica Bravo Gustavo Leone Peter Houghton Periannan Kuppusamy David E. Cohn Karuppaiyah Selvendiran

STAT3 iswell corroborated preclinically as a cancer therapeutic target, but tractable translational strategies for its blockade by small molecule inhibitors have remained elusive. In this study, we report the development of a novel class of bifunctional STAT3 inhibitors, based on conjugation of a diarylidenyl-piperidone (DAP) backbone to an N-hydroxypyrroline (–NOH) group, which exhibits minima...

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