نتایج جستجو برای: daminozide

تعداد نتایج: 69  

2009
Dmitry Miroshnichenko Mikhail Filippov Sergey Dolgov

The influence of daminozide, an inhibitor of gibberellins biosynthesis, on the somatic embryogenesis in immature and mature embryo derived from tissue cultures of wheat was investigated. Low concentrations of daminozide (0.064-0.127 mM) positively affected the somatic embryogenic capacity of immature embryos (cv. ‘Andros’) cultured on the medium supplemented with either 2,4-dichlorophenoxyaceti...

Journal: :Journal of medicinal chemistry 2012
Nathan R Rose Esther C Y Woon Anthony Tumber Louise J Walport Rasheduzzaman Chowdhury Xuan Shirley Li Oliver N F King Clarisse Lejeune Stanley S Ng Tobias Krojer Mun Chiang Chan Anna M Rydzik Richard J Hopkinson Ka Hing Che Michelle Daniel Claire Strain-Damerell Carina Gileadi Grazyna Kochan Ivanhoe K H Leung James Dunford Kar Kheng Yeoh Peter J Ratcliffe Nicola Burgess-Brown Frank von Delft Susanne Muller Brian Marsden Paul E Brennan Michael A McDonough Udo Oppermann Robert J Klose Christopher J Schofield Akane Kawamura

The JmjC oxygenases catalyze the N-demethylation of N(ε)-methyl lysine residues in histones and are current therapeutic targets. A set of human 2-oxoglutarate analogues were screened using a unified assay platform for JmjC demethylases and related oxygenases. Results led to the finding that daminozide (N-(dimethylamino)succinamic acid, 160 Da), a plant growth regulator, selectively inhibits the...

Journal: :Inorganics (Basel) 2023

Daminozide, a plant growth regulator, is an effective inhibitor of the Jumonji domain-containing protein (JMJD) histone demethylase. Herein, four ruthenium(II)/rhenium(I)-daminozide conjugates, with molecular formulas [Ru(N-N)2bpy(4-CH2OH-4′-CH2O-daminozide)](PF6)2 (Ru-1/Ru-2) (N-N = 1,10-phenanthroline (phen, in Ru-1) and 4,7-diphenyl-1,10-phenanthroline (DIP, Ru-2)) Re(N-N)(CO)3(PyCH2O-damino...

Ali Mohammadi Torkashvand Behzad Kaviani Davood Hashemabadi Shahram Shoa Kazemi

Pot marigold (Calendula officinalis L.) is a medicinal and ornamental plant. The effect of different concentrations of chlormequat (cycocel), and daminozide, two plant growth retardant, on plant height, flowering, the content of essence and some other traits in pot marigold (Calendula officinalis) was assessed. Plant growth retardants are commonly applied to limit stem elongation and produce a ...

Journal: :journal of ornamental plants 2014
shahram shoa kazemi davood hashemabadi ali mohammadi torkashvand behzad kaviani

pot marigold (calendula officinalis l.) is a medicinal and ornamental plant. the effect of different concentrations of chlormequat (cycocel), and daminozide, two plant growth retardant, on plant height, flowering, the content of essence and some other traits in pot marigold (calendula officinalis) was assessed. plant growth retardants are commonly applied to limit stem elongation and produce a ...

2015
Wenhui Gan Tom Bond Xin Yang Paul Westerhoff

1 N-nitrosodimethylamine (NDMA) is an emerging disinfection by-product, and we show 2 that use of chlorine dioxide (ClO2) has the potential to increase NDMA formation in waters 3 containing precursors with hydrazine moieties. NDMA formation was measured after 4 oxidation of 13 amines by monochloramine, ClO2 and pre-treatment with ClO2 followed by 5 post-monochloramination. Daminozide, a plant g...

2016
Jing-Yi Chen Chien-Feng Li Pei-Yi Chu You-Syuan Lai Chung-Hsing Chen Shih Sheng Jiang Ming-Feng Hou Wen-Chun Hung

Alterations of histone methylation dynamically regulated by methyltransferases and demethylases are frequently found in human cancers. Here, we showed that expression of lysine demethylase 2A (KDM2A) is markedly increased in human breast cancer and its overexpression is associated with tumor progression and poor prognosis. Knockdown of KDM2A in breast cancer cells reduced proliferation but not ...

Journal: :Mutagenesis 2010
David Kirkland Paul Fowler

In the analysis by Parry et al. [Parry, J. M., Parry, E., Phrakonkham, P. and Corvi, R. (2010) Analysis of published data for top concentration considerations in mammalian cell genotoxicity testing. Mutagenesis, 25, 531-538], 24 rodent carcinogens that were negative in the Ames test were identified that were only positive in mammalian cell tests at concentrations between 1 and 10 mM. These carc...

Journal: :Fundamental and applied toxicology : official journal of the Society of Toxicology 1988
P Sagelsdorff W K Lutz C Schlatter

[methyl-14C]Daminozide (succinic acid 2',2'-dimethylhydrazide; 37 mg/kg), 1,1-[14C]dimethylhydrazine (UDMH; 19 mg/kg), and [14C]dimethylnitrosamine (DMNA; 0.1 mg/kg) were administered by oral gavage to male Sprague-Dawley rats. After 24 hr, the animals were killed and DNA was purified from the livers to constant specific radioactivity. After enzymatic degradation of the DNA to the 3'-deoxynucle...

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