Somenewtriethylammoniumsalts,namelytriethylammonium4-(cyclohexyl-amino)-4-oxobut-2-enoate(B1),triethylammonium5-(cyclohexylamino)-5-oxopentanoate(B2),triethylammonium4-(cyclohexylamino)-4-oxobutanoate(B3)weresynthesizedasacorrosioninhibitorformildsteel.Thesesaltscouldtestinonemolaritysulfuricacidatroomtemperaturefor24hoursbyusingweightoflosingmethod.Theresultsrevealedthattheefficiencyofinhibiti...

5,981,180 A 11/1999 Chandleret a1. 6,046,807 A 4/2000 Chandler 6,139,800 A 10/2000 Chandler 6,268,222 B1 7/2001 Chandleret a1. 6,366,354 B1 4/2002 Chandler 6,449,562 B1 9/2002 Chandler et a1. 6,514,295 B1 2/2003 Chandleret a1. 6,524,793 B1 2/2003 Chandleret a1. 6,592,822 B1 7/2003 Chandler 6,599,331 B2 7/2003 Chandleret a1. 6,632,526 B1 10/2003 Chandler 6,649,414 B1 11/2003 Chandler et a1. 6,69...

In the course of screening for novel anticancer compounds, B1 [N-(2-(dimethylamino)ethyl)-2-aminothiazonaphthalimide], a novel amonafide analogue, was generated as a new anticancer candidate. In the present study, B1 displayed stronger antitumor effects than amonafide in HL60 cells. We further examined whether B1 overcomes the resistance conferred by Bcl-2, as overcoming the resistance conferre...

Lenstra, Lenstra, and Lovász in [7] proved several inequalities showing that the vectors in an LLL-reduced basis are short, and near orthogonal. Here we present generalizations, from which with k = 1, and k = n we can recover their inequalities: Theorem 1. Let b1, . . . , bn ∈ R be an LLL-reduced basis of the lattice L, and d1, . . . , dk arbitrary linearly independent vectors in L. Then ‖b1 ‖ ...

Chemotherapeutic drugs ideally should take advantage of the differences between transformed and normal cells and induce apoptosis only in cancer cells. One such difference may be the overexpression of cyclin B1 protein in cancer cells, which is required for the proper progression through mitosis. Previously, we showed that treatment of human prostate cancer cells with 2-methoxyestradiol (2-ME) ...

6,123,819 A * 9/2000 Peeters ....................... 204/452 6,361,958 B1 * 3/2002 Shieh et al. ................. 435/7.1 6,524,790 B1 * 2/2003 Kopf-Sill et al. .............. 435/6 6,585,939 B1 7/2003 Dapprich 6,599,436 B1 7/2003 Matzke et al. 6,613,512 B1 9/2003 Kopf-Sill et al. 6,649,358 B1 * 11/2003 Parce et al. .................. 435/7.2 6,699,665 B1 * 3/2004 Kim et al. ......................

Bradykinin (BK) and its receptors (B1 and B2 receptors) play important roles in inflammatory nociception. However, the patterns of expression and physiological/pathological functions of B1 and B2 receptors in trigeminal ganglion (TG) neurons remain to be fully elucidated. We investigated the functional expression of BK receptors in rat TG neurons. We observed intense immunoreactivity of B2 rece...