نتایج جستجو برای: 0632 and 056

تعداد نتایج: 16827472  

Journal: :Molecular pharmacology 2015
Maoqing Dong Ashton M Vattelana Polo C-H Lam Andrew J Orry Ruben Abagyan Arthur Christopoulos Patrick M Sexton David R Haines Laurence J Miller

Understanding the molecular basis of ligand binding to receptors provides insights useful for rational drug design. This work describes development of a new antagonist radioligand of the type 1 cholecystokinin receptor (CCK1R), (2-fluorophenyl)-2,3-dihydro-3-[(3-isoquinolinylcarbonyl)amino]-6-methoxy-2-oxo-l-H-indole-3-propanoate (T-0632), and exploration of the molecular basis of its binding. ...

Journal: :Bioorganic & medicinal chemistry 2010
Minsun Chang Seol-Rin Park Juhyun Kim Mijung Jang Jeong Hyun Park Ji Eun Park Hyeung-Geun Park Young-Ger Suh Yeon Su Jeong Young-Ho Park Hee-Doo Kim

In searching for opportunities to exploit the benefits of silicon in TRPV1 research, we tried to investigate the pharmacological effects of sila-substitution (C/Si exchange) of tert-butyl group in the MK-056 series. Compound 13a, with a 4-positioned trimethylsilanyl group on the B ring in place of tert-butyl group, exhibited the most potent antagonist activity with IC(50) values of 0.15 microM,...

2010
Sébastien Villéger Julia Ramos Miranda Domingo Flores Hernández

2013
Narasimha Murthy

*Corresponding Author: Dr. Srinivas. C, Department of Microbiology and Biotechnology, Bangalore University, Jnanabharathi Campus, Bangalore-560 056, Karnataka, India. Page| 342 Efficacy of Trichoderma asperellum against Ralstonia solanacearum under greenhouse conditions Narasimha Murthy K, Nirmala Devi D and Srinivas C* Department of Microbiology and Biotechnology, Bangalore University, Jnanabh...

Journal: :Publications of the Astronomical Society of Australia 2015

2012
S. M. Oliveira N. J. Teixeira L. Fernandes

S. M. Oliveira Faculdade de Ciências Médicas, Universidade Nova de Lisboa, Campo Mártires da Pátria, 130, 1169-056 Lisbon, Portugal and MedicalConsult, SA, Campo Grande, 56-88A, 1700-093 Lisbon, Portugal N. J. Teixeira Faculdade de Ciências Médicas, Universidade Nova de Lisboa, Campo Mártires da Pátria, 130, 1169-056 Lisbon, Portugal and Escola Superior de Tecnologia da Saúde de Lisboa, Institu...

Journal: :Pediatric Critical Care Medicine 2018

Journal: :Developmental and comparative immunology 2016
Yosra Ben Cheikh Marie-Agnès Travers Benjamin Morga Yoann Godfrin Damien Rioult Frank Le Foll

Bacterial isolates were obtained from mortality events affecting Mytilus edulis and reported by professionals in 2010-2013 or from mussel microflora. Experimental infections allowed the selection of two isolates affiliated to Vibrio splendidus/Vibrio hemicentroti type strains: a virulent 10/068 1T1 (76.6% and 90% mortalities in 24 h and 96 h) and an innocuous 12/056 M24T1 (0% and 23.3% in 24 h ...

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