نتایج جستجو برای: physicochemical property

تعداد نتایج: 188116  

Journal: :The Journal of General Physiology 1957
Roger M. Herriott James L. Barlow

A method of preparing the protein coats or ghosts of phage T2 is described along with proof that the lytic action is a property of the ghost. An assay based on the lytic action toward host cells has been developed which permits a rapid evaluation of the number of ghosts with a reliability of +/-15 per cent. The antigenic and certain physicochemical properties of the ghost have been determined.

2014
D Archana Laxmi Upadhyay Joydeep Dutta

Chitosan-pectin, chitosan-alginate and chitosan-pectin-alginate scaffolds were prepared by freeze-drying technique. The physicochemical characteristics of the scaffolds were characterized by FTIR and SEM. The biological activities like antibacterial assessment, swelling behavior, biodegradation and cytotoxicity study of the prepared scaffolds were evaluated. The results show high swelling prope...

2008
A. Saraswathy S. Nandini Devi D. Ramasamy

The ethanol crude extract of stem bark of Holoptelea integrifolia Planch. traditionally used in Indian system of medicine was screened for its antioxidant activity using α-tocopherol as standard antioxidant. The free radical scavenging potential of the extract was evaluated by two different antioxidant methods; ferric thiocyanate and thiobarbituric acid method. The ethanol extract was found to ...

2016
Aurélie Mallinger Kai Schiemann Christian Rink Frank Stieber Michel Calderini Simon Crumpler Mark Stubbs Olajumoke Adeniji-Popoola Oliver Poeschke Michael Busch Paul Czodrowski Djordje Musil Daniel Schwarz Maria-Jesus Ortiz-Ruiz Richard Schneider Ching Thai Melanie Valenti Alexis de Haven Brandon Rosemary Burke Paul Workman Trevor Dale Dirk Wienke Paul A. Clarke Christina Esdar Florence I. Raynaud Suzanne A. Eccles Felix Rohdich Julian Blagg

The Mediator complex-associated cyclin-dependent kinase CDK8 has been implicated in human disease, particularly in colorectal cancer where it has been reported as a putative oncogene. Here we report the discovery of 109 (CCT251921), a potent, selective, and orally bioavailable inhibitor of CDK8 with equipotent affinity for CDK19. We describe a structure-based design approach leading to the disc...

2014
Soo-Jin Choi Jin-Ho Choy

Biokinetic studies of zinc oxide (ZnO) nanoparticles involve systematic and quantitative analyses of absorption, distribution, metabolism, and excretion in plasma and tissues of whole animals after exposure. A full understanding of the biokinetics provides basic information about nanoparticle entry into systemic circulation, target organs of accumulation and toxicity, and elimination time, whic...

2012
Mingyun Shen Sheng Tian Youyong Li Qian Li Xiaojie Xu Junmei Wang Tingjun Hou

UNLABELLED BACKGROUND In this work, we analyzed and compared the distribution profiles of a wide variety of molecular properties for three compound classes: drug-like compounds in MDL Drug Data Report (MDDR), non-drug-like compounds in Available Chemical Directory (ACD), and natural compounds in Traditional Chinese Medicine Compound Database (TCMCD). RESULTS The comparison of the property ...

2008
Ravi Gupta Ankush Mittal Kuldip Singh

This paper presents a novel feature vector based on physicochemical property of amino acids for prediction protein structural classes. The proposed method is divided into three different stages. First, a discrete time series representation to protein sequences using physicochemical scale is provided. Later on, a wavelet-based time-series technique is proposed for extracting features from mapped...

2014
Kurt S. Van Horn Xiaohua Zhu Trupti Pandharkar Sihyung Yang Brian Vesely Manu Vanaerschot Jean-Claude Dujardin Suman Rijal Dennis E. Kyle Michael Zhuo Wang Karl A. Werbovetz Roman Manetsch

A series of N(2),N(4)-disubstituted quinazoline-2,4-diamines has been synthesized and tested against Leishmania donovani and L. amazonensis intracellular amastigotes. A structure-activity and structure-property relationship study was conducted in part using the Topliss operational scheme to identify new lead compounds. This study led to the identification of quinazolines with EC50 values in the...

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