نتایج جستجو برای: csf1

تعداد نتایج: 305  

Journal: :The New England journal of medicine 2015
William D Tap Zev A Wainberg Stephen P Anthony Prabha N Ibrahim Chao Zhang John H Healey Bartosz Chmielowski Arthur P Staddon Allen Lee Cohn Geoffrey I Shapiro Vicki L Keedy Arun S Singh Igor Puzanov Eunice L Kwak Andrew J Wagner Daniel D Von Hoff Glen J Weiss Ramesh K Ramanathan Jiazhong Zhang Gaston Habets Ying Zhang Elizabeth A Burton Gary Visor Laura Sanftner Paul Severson Hoa Nguyen Marie J Kim Adhirai Marimuthu Garson Tsang Rafe Shellooe Carolyn Gee Brian L West Peter Hirth Keith Nolop Matt van de Rijn Henry H Hsu Charles Peterfy Paul S Lin Sandra Tong-Starksen Gideon Bollag

BACKGROUND Expression of the colony-stimulating factor 1 (CSF1) gene is elevated in most tenosynovial giant-cell tumors. This observation has led to the discovery and clinical development of therapy targeting the CSF1 receptor (CSF1R). METHODS Using x-ray co-crystallography to guide our drug-discovery research, we generated a potent, selective CSF1R inhibitor, PLX3397, that traps the kinase i...

2015
Bin-Zhi Qian Hui Zhang Jiufeng Li Tianfang He Eun-Jin Yeo Daniel Y.H. Soong Neil O. Carragher Alison Munro Alvin Chang Anne R. Bresnick Richard A. Lang Jeffrey W. Pollard

Although the link between inflammation and cancer initiation is well established, its role in metastatic diseases, the primary cause of cancer deaths, has been poorly explored. Our previous studies identified a population of metastasis-associated macrophages (MAMs) recruited to the lung that promote tumor cell seeding and growth. Here we show that FMS-like tyrosine kinase 1 (Flt1, also known as...

Journal: :The Journal of Experimental Medicine 2001
Elaine Y. Lin Andrew V. Nguyen Robert G. Russell Jeffrey W. Pollard

In human breast carcinomas, overexpression of the macrophage colony-stimulating factor (CSF-1) and its receptor (CSF-1R) correlates with poor prognosis. To establish if there is a causal relationship between CSF-1 and breast cancer progression, we crossed a transgenic mouse susceptible to mammary cancer with mice containing a recessive null mutation in the CSF-1 gene (Csf1(op)) and followed tum...

Journal: :Journal of cell science 2008
Evangelia A Papakonstanti Olivier Zwaenepoel Antonio Bilancio Emily Burns Gemma E Nock Benjamin Houseman Kevan Shokat Anne J Ridley Bart Vanhaesebroeck

The class IA isoforms of phosphoinositide 3-kinase (p110alpha, p110beta and p110delta) often have non-redundant functions in a given cell type. However, for reasons that are unclear, the role of a specific PI3K isoform can vary between cell types. Here, we compare the relative contributions of PI3K isoforms in primary and immortalised macrophages. In primary macrophages stimulated with the tyro...

Journal: :Cell 2014
Paul Andrew Muller Balázs Koscsó Gaurav Manohar Rajani Korey Stevanovic Marie-Luise Berres Daigo Hashimoto Arthur Mortha Marylene Leboeuf Xiu-Min Li Daniel Mucida E. Richard Stanley Stephanie Dahan Kara Gross Margolis Michael David Gershon Miriam Merad Milena Bogunovic

Intestinal peristalsis is a dynamic physiologic process influenced by dietary and microbial changes. It is tightly regulated by complex cellular interactions; however, our understanding of these controls is incomplete. A distinct population of macrophages is distributed in the intestinal muscularis externa. We demonstrate that, in the steady state, muscularis macrophages regulate peristaltic ac...

2016
Adam R. Wolfe Nicholaus J Trenton Bisrat G. Debeb Richard Larson Brian Ruffell Khoi Chu Walter Hittelman Michael Diehl Jim M Reuben Naoto T. Ueno Wendy A. Woodward

Inflammatory breast cancer (IBC) is a unique and deadly disease with unknown drivers. We hypothesized the inflammatory environment contributes to the IBC phenotype. We used an in vitro co-culture system to investigate interactions between normal and polarized macrophages (RAW 264.7 cell line), bone-marrow derived mesenchymal stem cells (MSCs), and IBC cells (SUM 149 and MDA-IBC3). We used an in...

2013
Clare Pridans Kristin A. Sauter Kristin Baer Holger Kissel David A. Hume

Hereditary diffuse leukoencephalopathy with spheroids (HDLS) in humans is a rare autosomal dominant disease characterized by giant neuroaxonal swellings (spheroids) within the CNS white matter. Symptoms are variable and can include personality and behavioural changes. Patients with this disease have mutations in the protein kinase domain of the colony-stimulating factor 1 receptor (CSF1R) which...

2014
Larissa B. Patterson Emily J. Bain David M. Parichy

Fishes have diverse pigment patterns, yet mechanisms of pattern evolution remain poorly understood. In zebrafish, Danio rerio, pigment-cell autonomous interactions generate dark stripes of melanophores that alternate with light interstripes of xanthophores and iridophores. Here, we identify mechanisms underlying the evolution of a uniform pattern in D. albolineatus in which all three pigment ce...

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