نتایج جستجو برای: oxantel

تعداد نتایج: 32  

2014
Gordana Panic Urs Duthaler Benjamin Speich Jennifer Keiser

Helminth infections are responsible for a considerable public health burden, yet the current drug armamentarium is small. Given the high cost of drug discovery and development, the high failure rates and the long duration to develop novel treatments, drug repurposing circumvents these obstacles by finding new uses for compounds other than those they were initially intended to treat. In the pres...

Journal: :Molecular pharmacology 2010
Pingwei Zhao Haleli Sharir Ankur Kapur Alan Cowan Ellen B Geller Martin W Adler Herbert H Seltzman Patricia H Reggio Susanne Heynen-Genel Michelle Sauer Thomas D Y Chung Yushi Bai Wei Chen Marc G Caron Larry S Barak Mary E Abood

Known agonists of the orphan receptor GPR35 are kynurenic acid, zaprinast, 5-nitro-2-(3-phenylproplyamino) benzoic acid, and lysophosphatidic acids. Their relatively low affinities for GPR35 and prominent off-target effects at other pathways, however, diminish their utility for understanding GPR35 signaling and for identifying potential therapeutic uses of GPR35. In a screen of the Prestwick Li...

2016
Melanie Abongwa Samuel K Buxton Elise Courtot Claude L Charvet Cédric Neveu Ciaran J McCoy Saurabh Verma Alan P Robertson Richard J Martin

BACKGROUND AND PURPOSE Control of nematode parasite infections relies largely on anthelmintic drugs, several of which act on nicotinic ACh receptors (nAChRs), and there are concerns about the development of resistance. There is an urgent need for development of new compounds to overcome resistance and novel anthelmintic drug targets. We describe the functional expression and pharmacological cha...

Journal: :Antibiotics 2015
Jie Feng Megan Weitner Wanliang Shi Shuo Zhang David Sullivan Ying Zhang

Lyme disease is a leading vector-borne disease in the United States. Although the majority of Lyme patients can be cured with standard 2-4 week antibiotic treatment, 10%-20% of patients continue to suffer from prolonged post-treatment Lyme disease syndrome (PTLDS). While the cause for this is unclear, persisting organisms not killed by current Lyme antibiotics may be involved. In our previous s...

نمودار تعداد نتایج جستجو در هر سال

با کلیک روی نمودار نتایج را به سال انتشار فیلتر کنید