نتایج جستجو برای: propoxy

تعداد نتایج: 252  

Journal: :Acta Crystallographica Section E Structure Reports Online 2010

Journal: :Antimicrobial agents and chemotherapy 2005
C Ying A Holy D Hocková Z Havlas E De Clercq J Neyts

Novel acyclic nucleoside phosphonates with a pyrimidine base preferentially containing an amino group at C-2 and C-4 and a 2-(phosphonomethoxy)ethoxy or (R)-2-(phosphonomethoxy)propoxy group at C-6 selectively inhibit the replication of wild-type and lamivudine-resistant hepatitis B viruses. The activity of the most potent compounds was comparable to that of adefovir.

2010
Payam Khazaeli Mamoud Reza Heidari Alireza Foroumadi Mehdi Kalati

Evaluation the antinociceptive and antiinflammatory effect, of new rigid, propoxy benzopyrane-3,4 Di-hydroxychalcone derivative by Hot-plate, Formaline and Plethysmography Payam Khazaeli, Mamoud Reza Heidari, Alireza Foroumadi, Mehdi Kalati From 1 International Congress on Neurobiology and Clinical Psychopharmacology and European Psychiatric Association Conference on Treatment Guidance Thessalo...

Journal: :Molecular pharmacology 2014
Marc Lamphier Wanjun Zheng Eicke Latz Mark Spyvee Hans Hansen Jeffrey Rose Melinda Genest Hua Yang Christina Shaffer Yan Zhao Yongchun Shen Carrie Liu Diana Liu Thorsten R Mempel Christopher Rowbottom Jesse Chow Natalie C Twine Melvin Yu Fabian Gusovsky Sally T Ishizaka

The discovery that circulating nucleic acid-containing complexes in the serum of autoimmune lupus patients can stimulate B cells and plasmacytoid dendritic cells via Toll-like receptors 7 and 9 suggested that agents that block these receptors might be useful therapeutics. We identified two compounds, AT791 {3-[4-(6-(3-(dimethylamino)propoxy)benzo[d]oxazol-2-yl)phenoxy]-N,N-dimethylpropan-1-amin...

Journal: :Chemical & pharmaceutical bulletin 2002
Jin-Cherng Lien Li-Jiau Huang Che-Ming Teng Jih-Pyang Wang Sheng-Chu Kuo

In our continuing search for novel antiplatelet, antiallergic, and antiinflammatory agents, 2-alkoxy derivatives of 1,4-naphthoquinone were prepared. Some of these compounds showed significant antiplatelet, antiallergic, and antiinflammatory activities. Among them, 2-propoxy-1,4-naphthoquinone and 2-butoxy-1,4-naphthoquinone exhibited potent inhibitory effect on neutrophil superoxide anion form...

2016
Camille D. Dago Estelle Messé Olivier Mignen Christophe Brigaudeau Jean-Pierre Bazureau

1-{β-[3-(4-Methoxy-phenyl)propoxy]-4-methoxyphenethyl}-1H-imidazole hydrochloride 7, or SKF-96365, was synthesized in four steps with an overall yield of 9%. The structure of 7 was confirmed by 1H-, 13C-NMR, HRMS, and elemental analysis. The intermediates 3 and 4 were also isolated and characterized by 1H-, 13C-NMR, and HRMS.

Journal: :Molecules 2006
Fang Liu Jing-wie He Zheng-mei Lin Jun-qi Ling De-min Jia

A new dimethacrylate monomer 9,9'-bis[4-(2'-hydroxy-3'-methacryloyloxy-propoxy)phenyl] fluorene (3) with a molecular weight of 634 was synthesized in 51.4% yield by addition of a glycidyl ether group to 9,9'-bis(4-hydroxyphenyl) fluorene (1) by the reaction of compound 1 with epichlorohydrin, and then introducing the methacrylate moiety by the reaction of the epoxy group with methacrylic acid. ...

Journal: :The Journal of antibiotics 1980
C Urakawa K Nakano R Imai

A facile alcoholysis of 7-methoxymitosanes and 5-methoxyindolequinone under basic conditions was discovered and a series of 7-alkoxymitosanes were synthesized from mitomycins A and B using this reaction. They showed strong antibacterial activity against various Gram-positive and Gram-negative bacteria and were potent inhibitors of cultivating HeLa S-3 cells in vitro. Among them, 7-n-propoxy-7-d...

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