نتایج جستجو برای: fgfr

تعداد نتایج: 1529  

2001
Patrick Auguste Demirkan B. Gürsel Sylvie Lemière Diana Reimers Pedro Cuevas Fernando Carceller James P. Di Santo Andreas Bikfalvi

We undertook a series of systematic studies to address the role of fibroblast growth factor/fibroblast growth factor receptor (FGF/FGFR) activity in tumor growth and angiogenesis. We expressed dominant-negative FGFR2 (FGFR2-DN) or FGFR1 (FGFR1-DN) in glioma C6 cells by using constitutive or tetracycline-regulated expression systems. Anchorage-dependent or independent growth was inhibited in FGF...

Journal: :Cancer research 2001
P Auguste D B Gürsel S Lemière D Reimers P Cuevas F Carceller J P Di Santo A Bikfalvi

We undertook a series of systematic studies to address the role of fibroblast growth factor/fibroblast growth factor receptor (FGF/FGFR) activity in tumor growth and angiogenesis. We expressed dominant-negative FGFR2 (FGFR2-DN) or FGFR1 (FGFR1-DN) in glioma C6 cells by using constitutive or tetracycline-regulated expression systems. Anchorage-dependent or independent growth was inhibited in FGF...

Journal: :Molecular cancer research : MCR 2010
Ellen Margrethe Haugsten Antoni Wiedlocha Sjur Olsnes Jørgen Wesche

The fibroblast growth factor receptors (FGFR) play essential roles both during development and in the adult. Upon ligand binding, FGFRs induce intracellular signaling networks that tightly regulate key biological processes, such as cell proliferation, survival, migration, and differentiation. Deregulation of FGFR signaling can thus alter tissue homeostasis and has been associated with several d...

Journal: :Investigative ophthalmology & visual science 2008
Sandrine Siffroi-Fernandez Marie-Paule Felder-Schmittbuhl Hemant Khanna Anand Swaroop David Hicks

PURPOSE Several fibroblast growth factors (FGFs) exhibit neuroprotective influences against retinal photoreceptor degeneration. The expression of FGF receptor (FGFR) 4 on photoreceptors suggests a specific ligand, FGF-19, might also be beneficial. The authors hence examined the potential role of FGF-19 in this regard. METHODS Adult human retinal sections were processed for anti-FGFR-4 immunoh...

Journal: :The Journal of biological chemistry 1994
M Roghani A Mansukhani P Dell'Era P Bellosta C Basilico D B Rifkin D Moscatelli

The role of heparin or heparan sulfates in the interaction of basic fibroblast growth factor (bFGF) with its high affinity receptor were investigated using purified extracellular ligand-binding region of FGF receptor-1 (FGFR-1) and intact receptors expressed in a myeloid cell line (32D) that does not express detectable levels of heparan sulfate proteoglycans or in Chinese hamster ovary (CHO) ce...

Journal: :Molecular cancer therapeutics 2015
Jae-Cheol Jo Eun Kyoung Choi Jae-Sik Shin Jai-Hee Moon Seung-Woo Hong Ha-Reum Lee Seung-Mi Kim Soo-A Jung Dae-Hee Lee Seang Hwan Jung Sun-Hye Lee Jeong Eun Kim Kyu-pyo Kim Yong Sang Hong Young-Ah Suh Se Jin Jang Eun Kyung Choi Jung Shin Lee Dong-Hoon Jin Tae Won Kim

The MET receptor tyrosine kinase, the receptor for hepatocyte growth factor (HGF), has been implicated in cancer growth, invasion, migration, angiogenesis, and metastasis in a broad variety of human cancers, including human hepatocellular carcinoma (HCC). Recently, MET was suggested to be a potential target for the personalized treatment of HCC with an active HGF-MET signaling pathway. However,...

Journal: :Clinical cancer research : an official journal of the American Association for Cancer Research 2017
Florian Malchers Meryem Ercanoglu Daniel Schütte Roberta Castiglione Verena Tischler Sebastian Michels Ilona Dahmen Johannes Brägelmann Roopika Menon Johannes M Heuckmann Julie George Sascha Ansén Martin L Sos Alex Soltermann Martin Peifer Jürgen Wolf Reinhard Büttner Roman K Thomas

Purpose: The 8p12-p11 locus is frequently amplified in squamous cell lung cancer (SQLC); the receptor tyrosine kinase fibroblast growth factor receptor 1 (FGFR1) being one of the most prominent targets of this amplification. Thus, small molecules inhibiting FGFRs have been employed to treat FGFR1-amplified SQLC. However, only about 11% of such FGFR1-amplified tumors respond to single-agent FGFR...

2016
Anna Szlachcic Malgorzata Zakrzewska Michal Lobocki Piotr Jakimowicz Jacek Otlewski

Fibroblast growth factor receptors (FGFRs) are attractive candidate cancer therapy targets as they are overexpressed in multiple types of tumors, such as breast, prostate, bladder, and lung cancer. In this study, a natural ligand of FGFR, an engineered variant of fibroblast growth factor 1 (FGF1V), was conjugated to a potent cytotoxic drug, monomethyl auristatin E (MMAE), and used as a targetin...

Journal: :Development 2005
Giuseppe Lupo Ying Liu Rong Qiu Roshantha A S Chandraratna Giuseppina Barsacchi Rong-Qiao He William A Harris

In the developing spinal cord and telencephalon, ventral patterning involves the interplay of Hedgehog (Hh), Retinoic Acid (RA) and Fibroblast Growth Factor (FGF) signaling. In the eye, ventral specification involves Hh signaling, but the roles of RA and FGF signaling are less clear. By overexpression assays in Xenopus embryos, we found that both RA and FGF receptor (FGFR) signaling ventralize ...

2016
Ying Lin Hongbin Gao Siming Ai Jacob V.P. Eswarakumar Tao Li Bingqian Liu Hongye Jiang Yuhua Liu Xialin Liu Yonghao Li Yao Ni Jiangna Chen Zhuoling Lin Xiaoling Liang Chenjin Jin Xinhua Huang Lin Lu Yizhi Liu

Crouzon syndrome, a dominantly inherited disorder and the most common type of craniosynostosis syndrome, is caused by mutations in the fibroblast growth factor receptor 2 (FGFR 2) gene, and characterized by craniosynostosis, shallow orbits, ocular proptosis, midface hypoplasia and a curved, beak‑like nose. The purpose of the present study was to investigate the fibroblast growth factor receptor...

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