SOME UNUSUAL REACTIONS OF 3-PHENYLAMINOISOXAZOL-5 (2H)- ONES
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Abstract:
3-Phenylaminoisoxazol-5(2H)-ones,s ubstituted on nitrogen with an isoquinoline or quinazoline group, react with tertiary amine bases to give imidazo annelated compounds. When the N-substituent is a nitropyridine, 2-aminoindole derivatives are formed instead. Evidence is presented that the reactions proceed by initial addition of the tertiary arnine to C-4
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Journal title
volume 11 issue 1
pages -
publication date 2000-03-01
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