Application of N-methylimidazole for the Synthesis of Dimethyl-{3-methyl-2-[(alkoxycarbonyl) anilino]-2,3-dihydro-1H-imidazol-1-yl)}-2-butenedioate Derivatives
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Abstract:
A one-pot synthesis ofdimethyl-{3-methyl-2-[(alkoxycarbonyl) anilino]-2,3-dihydro-1Himidazol-1-yl)}-2-butenedioatesanddimethyl-2-[(alkoxycarbonyl)anilino]-2-butenedioates derivatives via reactions between dimethyl acetylenedicarboxylate,1-methylimidazoleand N-phenylcarbamates is described. The mild reaction condition, simple mixing of the starting materials and good yields exhibit the synthetic advantage of this method.
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application of n-methylimidazole for the synthesis of dimethyl-{3-methyl-2-[(alkoxycarbonyl) anilino]-2,3-dihydro-1h-imidazol-1-yl)}-2-butenedioate derivatives
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Journal title
volume 8 issue 2
pages 71- 76
publication date 2014-11-01
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