Aquastatin A, an inhibitor of mammalian adenosine triphosphatases from Fusarium aquaeductuum. Taxonomy, fermentation, isolation, structure determination and biological properties.

نویسندگان

  • K Hamano
  • M Kinoshita-Okami
  • K Minagawa
  • H Haruyama
  • T Kinoshita
  • T Hosoya
  • K Furuya
  • K Kinoshita
  • K Tabata
  • A Hemmi
چکیده

A new inhibitor of mammalian adenosine triphosphatases, designated aquastatin A, has been isolated from a fungus identified as Fusarium aquaeductuum. The structure of this compound has been determined by MS and NMR analyses. It inhibits Na+/K(+)-ATPase with an IC50 value of 7.1 microM, and H+/K(+)-ATPase with an apparent IC50 value of 6.2 microM.

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عنوان ژورنال:
  • The Journal of antibiotics

دوره 46 11  شماره 

صفحات  -

تاریخ انتشار 1993