Iron-Catalyzed C H Fuctionalization of Indoles
نویسندگان
چکیده
An easily available iron catalyst was developed to accomplish the C H functionalization of indoles with a-aryl-a-diazoesters in high yields under mild conditions. The asymmetric C H functionalization of indoles was also realized by using iron complexes of chiral spiro bisoxazolines with up to 78% ee.
منابع مشابه
Preparation of indoles via iron catalyzed direct oxidative coupling.
Iron-catalyzed aryl C-H and vinyl C-H bonds activation to give valuable substituted indole products was reported. The reaction shows high functional group tolerance.
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