Identification of AICP as a GluN2C-selective NMDA receptor superagonist at the GluN1 glycine site
نویسندگان
چکیده
Department of Molecular Screening, H. Lundbeck A/S, Valby, Denmark (M.J., K.F., A.D.); Present Address: Clinical Development, Chr. Hansen A/S, Hørsholm, Denmark (A.D.); Department of Drug Design and Pharmacology, University of Copenhagen, Copenhagen, Denmark (M.J., R.P.C., H.B.-O.); Department of Medicinal Chemistry 1, H. Lundbeck A/S, Valby, Denmark (P.K.); and Department of Biomedical and Pharmaceutical Sciences, University of Montana, Missoula, Montana, USA (F.Y., K.B.H.) This article has not been copyedited and formatted. The final version may differ from this version. Molecular Pharmacology Fast Forward. Published on June 6, 2017 as DOI: 10.1124/mol.117.108944
منابع مشابه
Structural determinants and mechanism of action of a GluN2C-selective NMDA receptor positive allosteric modulator.
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