Semisynthesis and insecticidal activity of some novel fraxinellone-based thioethers containing 1,3,4-oxadiazole moiety
نویسندگان
چکیده
Two series of novel fraxinellone-based thioethers containing 1,3,4-oxadiazole moiety were prepared as insecticidal agents against the oriental armyworm, Mythimna separata Walker. The structural assignment was based on the spectroscopic and X-ray analysis data. Among all the target compounds, compounds 4b, 4k, 5b, 5j and 5k exhibited more potent insecticidal activity with final mortality rates (FMRs) of more than 65%, especially 4k with the FMR of 75.9%, when compared with toosendanin. Some interesting results of structure-activity relationships are also discussed.
منابع مشابه
New Thermally Stable Aromatic Polyimides Based on Aromatic Diamine 2,5-Bis(3-amino-4-methyl benzene)-1,3,4-oxadiazole (BAMO): Synthesis and Characterization
In current study, the synthesis and characterization of novel thermally stable polyimides (PIs) containing an 1,3,4-oxadiazole moiety based on a diamine, i.e. 2,5-bis(3-amino-4-methyl benzene)-1,3,4-oxadiazole (BAMO), have been reported. The polymers were characterized using FT-IR and elemental analysis (CHN). Thermal and mechanical behaviours of the prepared PIs were studied by thermo-gravimet...
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