Synthesis of functionalized tryptamines by Brønsted acid catalysed cascade reactions.

نویسندگان

  • Nicola Melis
  • Francesco Secci
  • Thomas Boddaert
  • David J Aitken
  • Angelo Frongia
چکیده

An original synthetic protocol has been developed for the preparation of highly functionalized tryptamines from 2-hydroxycyclobutanone and secondary arylamines via a solvent-free Brønsted acid catalysed two-step reaction sequence.

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عنوان ژورنال:
  • Chemical communications

دوره 51 83  شماره 

صفحات  -

تاریخ انتشار 2015