TDAE strategy for the synthesis of 2,3-diaryl N-tosylaziridines.
نویسندگان
چکیده
We report herein an original and rapid synthesis of 2,3-diaryl N-tosylaziridines by TDAE strategy starting from ortho- or para-nitro(dichloromethyl)benzene derivatives and N-tosylimines. A mixture of cis/trans isomers was isolated from 1-(dichloromethyl)-4-nitrobenzene, whereas only trans-aziridines were obtained from ortho-nitro derivatives.
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ورودعنوان ژورنال:
- Molecules
دوره 18 7 شماره
صفحات -
تاریخ انتشار 2013