Selective N-Benzylation of Amino Acids under Homogeneously Catalyzed Hydrogenation Conditions
نویسندگان
چکیده
منابع مشابه
Enantioselective synthesis of beta2-amino acids using rhodium-catalyzed hydrogenation.
A series of protected beta2-dehydroamino acids has been prepared in three steps from commercially available starting materials in good yields. These were used as substrates in rhodium-catalyzed asymmetric hydrogenation applying a mixed ligand system of monodentate phosphoramidites and phosphines. Optimization of the catalyst structure was achieved by high throughput experimentation. High enanti...
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ژورنال
عنوان ژورنال: Synlett
سال: 2004
ISSN: 0936-5214,1437-2096
DOI: 10.1055/s-2004-836043