Multicomponent reaction of benzyl halides: Synthesis of [1,2,4]triazolo/benzimidazolo quinazolinones
نویسندگان
چکیده
منابع مشابه
Imides: forgotten players in the Ugi reaction. One-pot multicomponent synthesis of quinazolinones.
Up to now, the synthesis of quinazolinones has required lengthy synthetic procedures. Here, we describe an innovative one-pot multicomponent reaction leading to highly substituted quinazolinones. We believe that this novel transformation may open the door for the generation of new and pharmacologically active quinazolinones, but, most important of all, the resurrection of the imide-Ugi scaffold...
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ژورنال
عنوان ژورنال: Synthetic Communications
سال: 2016
ISSN: 0039-7911,1532-2432
DOI: 10.1080/00397911.2016.1140784