Inability of Isoquinoline Derivatives to Inhibit Virus Neuraminidase Activity
نویسندگان
چکیده
منابع مشابه
Inability of isoquinoline derivatives to inhibit virus neuraminidase activity.
The Selective Release of Proteins from a Bovine Enterovirus. By S. J. MARTIN and M.D. JOHNSTON Haemagglutinin Relationships of Hong Kong(H3) and Asian(H2) Influenza Strains Delineated by Antigen-specific Recombinants. By W.R. DOWDLE, W. M. MA~NE, M. COLEMAN and V. KNEZ The Kinetics of Haemagglutination by Semliki Forest Virus: a New Sedimentation-enumeration Method. By K. R. CAMERON and C. J. B...
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1,3-Dipolar cycloaddition of azomethine ylides derived from acenaphthylene-1,2-dione and 5methyl-benzo[b]-thiophene-2,3-dione with L-proline, thiazolidine-4-carboxylic acid and 1,2,3,4tetrahydroisoquinoline-3-carboxylic acid with various electron deficient dipolarophiles leads to the formation of novel spiroheterocycles having two or more chiral centers. Semiempirical studies have been performe...
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The main objective of this work was to synthesize novel compounds with a benzo[de][1,2,4]triazolo[5,1-a]isoquinoline scaffold by employing (dioxo-benzo[de]isoquinolin-2-yl) thiourea as a building block. Molecular docking was conducted in the COX-2 active site to predict the plausible binding mode and rationalize the structure-activity relationship of the synthesized compounds. The structures of...
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Objective(s) Some properties of neuraminidase produced by Pseudomonas aeruginosa PAO1 growth in a defined medium (BHI) were examined and evaluated for its features. Materials and Methods The obtained supernatant enzyme of P. aeruginosa PAO1 cultures was used in a sensitive fluorometric assay by using 2'-(4-methylumbelliferyl) a-D-N acetylneuraminic acid as substrate. As hydrolyzing MUN with ...
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ژورنال
عنوان ژورنال: Journal of General Virology
سال: 1972
ISSN: 0022-1317,1465-2099
DOI: 10.1099/0022-1317-16-2-227