Copper-Catalyzed Direct Benzylation ofβ-Ketoesters withN-Tosylhydrazones
نویسندگان
چکیده
منابع مشابه
Copper-catalyzed N-alkylation of indoles by N-tosylhydrazones
An efficient method for the direct N-alkylation of indoles via copper-catalyzed reductive cross coupling between N-tosylhydrazones and indole reagents has been developed. The reaction was performed in the presence of copper iodide and potassium hydroxide by utilization of tri(p-tolyl)phosphine as a ligand. A wide variety of N-alkylated indoles were obtained in moderate to good yields. The appli...
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ژورنال
عنوان ژورنال: Chinese Journal of Organic Chemistry
سال: 2015
ISSN: 0253-2786
DOI: 10.6023/cjoc201410045