نتایج جستجو برای: α-MSH

تعداد نتایج: 166080  

Journal: :Antimicrobial agents and chemotherapy 2011
Madhuri Singh Kasturi Mukhopadhyay

Alpha-melanocyte-stimulating hormone (α-MSH) is an endogenous neuropeptide that is known for its anti-inflammatory and antipyretic activities. We recently demonstrated that α-MSH possesses staphylocidal activity and causes bacterial membrane damage. To understand the role of its amino acid sequences in the staphylocidal mechanism, in the present study we investigated the antimicrobial activitie...

Journal: :iranian journal of pharmaceutical research 0
danial shamshirian department of radiopharmacy, school of pharmacy, tehran university of medical sciences, tehran, iran mostafa erfani radiation application research school, nuclear science and technology research institute (nstri), tehran, iran davood beiki research center for nuclear medicine, tehran university of medical sciences, tehran, iran maliheh hajiramazanali department of radiopharmacy, school of pharmacy, tehran university of medical sciences, tehran, iran. babak fallahi research center for nuclear medicine, tehran university of medical sciences, tehran, iran

melanocortin-1 (mc1) receptor is an attractive melanoma-specific target for the development of α-msh peptide based imaging and therapeutic agents. in this work a new lactam bridge α-msh analogue was synthesized and radiolabeled with 99mtc via hynic chelator and tricine as co-ligand. also, stability in human serum, receptor bound internalization and tissue biodistribution in tumor bearing nude m...

2018
Kathleen G. Mountjoy Alexandre Caron Kristina Hubbard Avik Shome Angus C. Grey Bo Sun Sarah Bould Martin Middleditch Beau Pontré Ailsa McGregor Paul W.R. Harris Renata Kowalczyk Margaret A. Brimble Rikus Botha Karen M.L. Tan Sarah J. Piper Christina Buchanan Syann Lee Anthony P. Coll Joel K. Elmquist

OBJECTIVE Regulation of energy balance depends on pro-opiomelanocortin (POMC)-derived peptides and melanocortin-4 receptor (MC4R). Alpha-melanocyte stimulating hormone (α-MSH) is the predicted natural POMC-derived peptide that regulates energy balance. Desacetyl-α-MSH, the precursor for α-MSH, is present in brain and blood. Desacetyl-α-MSH is considered to be unimportant for regulating energy b...

2017
Hong-Zai Guan Jing Dong Zheng-Yao Jiang Xi Chen

Alpha-melanocyte-stimulating hormone (α-MSH) is processed from proopiomelanocortin (POMC) and acts on the melanocortin receptors, MC3 and MC4. α-MSH plays a key role in energy homeostasis. In the present study, to shed light on the mechanisms by which α-MSH exerts its anorectic effects, extracellular neuronal activity was recorded in the hypothalamus and the dorsal vagal complex (DVC) of anesth...

2014
Jiun-Han Chen Junn-Liang Chang Pei-Ru Chen Yun-Ju Chuang Shih-Tsang Tang Shwu-Fen Pan Tzer-Bin Lin Kang-Hua Chen Mei-Jung Chen

The purpose of this study was to investigate if PPARγ plays a role in the melanogenesis. B16/F10 cells were divided into five groups: control, melanin stimulating hormone (α-MSH), α-MSH+retinol, α-MSH+GW9662 (PPARγ antagonist), and GW9662. Cells in the control group were cultured in the Dulbecco's modified Eagle's medium (DMEM) for 48 hrs. To initiate the melanogenesis, cells in all α-MSH group...

Journal: :Stroke 2011
Dannielle Zierath Pat Tanzi Kevin Cain Dean Shibata Kyra Becker

BACKGROUND AND PURPOSE α-Melanocyte stimulating hormone (α-MSH) is an endogenously produced neuropeptide derived from the same precursor as adrenocorticotropic hormone. α-MSH has profound immunomodulatory properties and may also be neuroprotective. Nothing is known about α-MSH and changes in its plasma concentrations in patients with acute ischemic stroke. METHODS In this prospective observat...

Ahmad Zare Shahneh JM Gooden Khatereh Bolouri Oskoui Navid Dadashpour Davachi Peter Wynn

  Background:Chronic active adrenocorticotropin hormone (ACTH) immunization of ewes (with a previous history of immunization) resulted in elevated titres of antibody against ACTH, which induced a reduction in circulating levels of cortisol. Objectives:<span style="color: win...

2013
Madhuri Singh Ravisekhar Gadepalli Benu Dhawan Kasturi Mukhopadhyay

Our previous studies revealed that alpha-melanocyte stimulating hormone (α-MSH) is strongly active against Staphylococcus aureus (S. aureus) including methicillin resistant S. aureus (MRSA). Killing due to α-MSH occurred by perturbation of the bacterial membrane. In the present study, we investigated the in vitro synergistic potential of α-MSH with five selected conventional antibiotics viz., o...

2013
Petteri Rinne Anna-Maija Penttinen Wendy Nordlund Markku Ahotupa Eriika Savontaus

Melanocyte-stimulating hormones, α-, β- and γ-MSH, regulate important physiological functions including energy homeostasis, inflammation and sodium metabolism. Previous studies have shown that α-MSH increases sodium excretion and promotes vascular function in rodents, but it is unexplored whether these characteristics of α-MSH could translate into therapeutic benefits in the treatment of hypert...

2016
Lu Gan Zhenjiang Liu Yizhe Chen Dan Luo Fei Feng Guannv Liu Chao Sun

Alpha melanocyte stimulating hormone (α-MSH) and Forkhead box C2 protein (Foxc2) enhance lipolysis in multiple tissues. However, their relationship in adipose fatty acid oxidation (FAO) remains unclear. Here, we demonstrated that α-MSH and Foxc2 increased palmitate oxidation to CO2 in white (WAT) and brown adipose tissue (BAT). C/EBPβ expression was reduced by α-MSH and Foxc2. FFA level was ele...

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