نتایج جستجو برای: hantzsch method

تعداد نتایج: 1630350  

A simple and mild one-pot three-component reaction for the preparation 1,4-dihydropyridines has been developed from various aldehyde substrates, 1,3-dicarbonyl compounds (dimedone) and ammonium acetate (Hantzsch method) in the presence of a catalytic amount of phospho sulfonic acid (PSA) as an efficient and heterogeneous solid acid in EtOH at room temperature. Preparation of PSA is straightforw...

2000
Andrea Arany Otto Meth-Cohn Miklós Nyerges

A variety of novel ligands have been generated by Vilsmeier formylation of Hantzsch pyridines. These compounds which we call DOTTADs contain two aldehyde, imine or amine functions flanking a central pyridine nitrogen and can be homochiral or crown derivatives. The synthesis and manipulation of these systems is discussed. © 2000 Elsevier Science Ltd. All rights reserved. Some years ago we descri...

A simple and mild one-pot three-component reaction for the preparation 1,4-dihydropyridines has been developed from various aldehyde substrates, 1,3-dicarbonyl compounds (dimedone) and ammonium acetate (Hantzsch method) in the presence of a catalytic amount of phospho sulfonic acid (PSA) as an efficient and heterogeneous solid acid in EtOH at room temperature. Preparation of PSA is straightforw...

Journal: :Molecules 2013
Adriana Ignat Ignat Grozav Luiza Gaina Victor Kuete Luminita Silaghi-Dumitrescu Thomas Efferth Valentin Zaharia

New aryl-hydrazinyl-1,3-selenazole and aroyl-hydrazonyl-1,3-selenazoles were synthesized via Hantzsch type condensation reactions of selenosemicarbazides with α-halogenocarbonyl derivatives, under classical versus microwave heating conditions. Excellent yields and shorter reaction times were obtained under irradiation conditions. The structures of the synthesized compounds were assigned based o...

Journal: :Organic letters 2014
Zhengxu S Han Yibo Xu Daniel R Fandrick Sonia Rodriguez Zhibin Li Bo Qu Nina C Gonnella Sanjit Sanyal Jonathan T Reeves Shengli Ma Nelu Grinberg Nizar Haddad Dhileep Krishnamurthy Jinhua J Song Nathan K Yee Waldemar Pfrengle Markus Ostermeier Jürgen Schnaubelt Zeno Leuter Sonja Steigmiller Jürgen Däubler Emanuel Stehle Lukas Neumann Thomas Trieselmann Patrick Tielmann Annette Buba Rainer Hamm Gunter Koch Svenja Renner Juan R Dehli Florian Schmelcher Christian Stange Jürgen Mack Rainer Soyka Chris H Senanayake

An efficient enantioselective synthesis of the chiral polycyclic cholesteryl ester transfer protein (CETP) inhibitor 1 has been developed. The synthesis was rendered practical for large scale via the development of a modified Hantzsch-type reaction to prepare the sterically hindered pyridine ring, enantioselective hydrogenation of hindered ketone 6 utilizing novel BIBOP-amino-pyridine derived R...

Journal: :journal of sciences islamic republic of iran 0

hantzsch 1,4-dihydropyridines are oxidized to the corresponding pyridine derivatives using oxygen or air and a mixture of the manganese and cobalt salts of parninobenzoic acid supported on silica gel as the catalysts. reactions are clean and the catalysts can be recovered easily and reused repeatedly.

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