نتایج جستجو برای: reactivators

تعداد نتایج: 133  

Journal: :Chemical research in toxicology 2010
Apurba K Bhattacharjee Kamil Kuca Kamil Musilek Richard K Gordon

Organophosphorus (OP) nerve agents that inhibit acetylcholinesterase (AChE; EC 3.1.1.7) function in the nervous system, causing acute intoxication. If untreated, death can result. Inhibited AChE can be reactivated by oximes, antidotes for OP exposure. However, OP intoxication caused by the nerve agent tabun (GA) is particularly resistant to oximes, which poorly reactivate GA-inhibited AChE. In ...

Journal: :Protein science : a publication of the Protein Society 2011
Benoît Sanson Jacques-Philippe Colletier Yechun Xu P Therese Lang Hualiang Jiang Israel Silman Joel L Sussman Martin Weik

The transient opening of a backdoor in the active-site wall of acetylcholinesterase, one of nature's most rapid enzymes, has been suggested to contribute to the efficient traffic of substrates and products. A crystal structure of Torpedo californica acetylcholinesterase in complex with the peripheral-site inhibitor aflatoxin is now presented, in which a tyrosine at the bottom of the active-site...

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