نتایج جستجو برای: dgat2 mogat2

تعداد نتایج: 161  

Journal: :Biotechnology for Biofuels 2021

Abstract Background Lipid transporters play an essential role in lipid delivery and distribution, but their influence on seed oil production oilseed crops is not well studied. Results Here, we examined the effect of two transporters, FAX1 ( fatty acid export1 ) ABCA9 ATP-binding cassette transporter subfamily A9 metabolism plant Camelina sativa . Overexpression (OE) increased weight size, with ...

2002
Hubert C. Chen Steven J. Smith Zuleika Ladha Dalan R. Jensen Luis D. Ferreira Leslie K. Pulawa James G. McGuire Robert E. Pitas Robert H. Eckel Robert V. Farese

Because obesity results from an imbalance between energy input and output, with most of the excess calories stored as triglycerides (or triacylglycerols), inhibition of triglyceride synthesis may prevent or reverse obesity (1). One of the key enzymes in triglyceride synthesis is acyl coenzyme A:diacylglycerol acyltransferase (acyl CoA:diacylglycerol acyltransferase, or DGAT), which catalyzes th...

Journal: :Journal of medicinal chemistry 2015
Kentaro Futatsugi Daniel W Kung Suvi T M Orr Shawn Cabral David Hepworth Gary Aspnes Scott Bader Jianwei Bian Markus Boehm Philip A Carpino Steven B Coffey Matthew S Dowling Michael Herr Wenhua Jiao Sophie Y Lavergne Qifang Li Ronald W Clark Derek M Erion Kou Kou Kyuha Lee Brandon A Pabst Sylvie M Perez Julie Purkal Csilla C Jorgensen Theunis C Goosen James R Gosset Mark Niosi John C Pettersen Jeffrey A Pfefferkorn Kay Ahn Bryan Goodwin

The medicinal chemistry and preclinical biology of imidazopyridine-based inhibitors of diacylglycerol acyltransferase 2 (DGAT2) is described. A screening hit 1 with low lipophilic efficiency (LipE) was optimized through two key structural modifications: (1) identification of the pyrrolidine amide group for a significant LipE improvement, and (2) insertion of a sp(3)-hybridized carbon center in ...

Journal: :The Journal of biological chemistry 2014
Jun Zhang Dan Xu Jia Nie Jingsong Cao Yonggong Zhai Dewen Tong Yuguang Shi

Acyl-CoA:monoacylglycerol acyltransferases (MGATs) and diacylglycerol acyltransferases (DGATs) catalyze the two consecutive steps in the synthesis of triacylglycerol, a key process required for dietary fat absorption into the enterocytes of the small intestine. In this report, we investigated the tendency of MGAT2 to form an enzyme complex with DGAT1 and DGAT2 in intact cells. We demonstrated t...

2017
Ling Zheng Jay Shockey Fei Bian Gao Chen Lei Shan Xinguo Li Shubo Wan Zhenying Peng

Diacylglycerol acyltransferase (DGAT) catalyzes the final step in triacylglycerol (TAG) biosynthesis via the acyl-CoA-dependent acylation of diacylglycerol. This reaction is a major control point in the Kennedy pathway for biosynthesis of TAG, which is the most important form of stored metabolic energy in most oil-producing plants. In this study, Arachis hypogaea type 2 DGAT (AhDGAT2) genes wer...

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