نتایج جستجو برای: auto inhibition

تعداد نتایج: 354924  

2015
Kevin Wu

OpenTuner can help users achieve better or more portable performance in their speci c domain through program autotuning. A key challenge for users seeking good autotuning performance in OpenTuner is selecting a search approach appropriate for problem. However, not only are current in-situ learning search approaches not robust enough to handle all search spaces, but there are also too many possi...

2014
Meike Bechtold Jörg Schultz Sven Bogdan

Eukaryotic cells have evolved a variety of actin-binding proteins to regulate the architecture and the dynamics of the actin cytoskeleton in time and space. The Diaphanous-related formins (DRF) represent a diverse group of Rho-GTPase-regulated actin regulators that control a range of actin structures composed of tightly-bundled, unbranched actin filaments as found in stress fibers and in filopo...

2012
Jing Xu Babu J. N. Reddy Preetha Anand Zhanyong Shu Silvia Cermelli Michelle K. Mattson Suvranta K. Tripathy Matthew T. Hoss Nikita S. James Stephen J. King Lan Huang Lee Bardwell Steven P. Gross

Kinesin-1 is a plus-end microtubule-based motor, and defects in kinesin-based transport are linked to diseases including neurodegeneration. Kinesin can auto-inhibit via a head-tail interaction, but is believed to be active otherwise. Here we report a tail-independent inactivation of kinesin, reversible by the disease-relevant signalling protein, casein kinase 2 (CK2). The majority of initially ...

2018
Ryuta Asaumi Kota Toshimoto Yoshifusa Tobe Kenta Hashizume Ken‐ichi Nunoya Haruo Imawaka Wooin Lee Yuichi Sugiyama

This study aimed to construct a physiologically based pharmacokinetic (PBPK) model of rifampicin that can accurately and quantitatively predict complex drug-drug interactions (DDIs) involving its saturable hepatic uptake and auto-induction. Using in silico and in vitro parameters, and reported clinical pharmacokinetic data, rifampicin PBPK model was built and relevant parameters for saturable h...

2017
Andrew Santiago-Frangos Jeliazko R Jeliazkov Jeffrey J Gray Sarah A Woodson

The RNA chaperone Hfq is an Sm protein that facilitates base pairing between bacterial small RNAs (sRNAs) and mRNAs involved in stress response and pathogenesis. Hfq possesses an intrinsically disordered C-terminal domain (CTD) that may tune the function of the Sm domain in different organisms. In Escherichia coli, the Hfq CTD increases kinetic competition between sRNAs and recycles Hfq from th...

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