نتایج جستجو برای: alisertib

تعداد نتایج: 124  

2018
Alexander Baumann Anna Maria S. Buchberger Guido Piontek Dominik Schüttler Martina Rudelius Rudolf Reiter Lena Gebel Gerhard Piendl Gero Brockhoff Anja Pickhard

Recently the Aurora-Kinases (Aurk) moved into the focus as novel disease related biomarkers and therapeutic targets. Elevated Aurora-Kinase expression has been found in a number of malignancies, amongst them HNSCC. For esophageal cancer, the AurkA Phe31-Ile polymorphism has previously been associated with tumor progression. Here we evaluated the treatment efficiency of HNSCC cell radiation as a...

2017
Mateusz Opyrchal Malgorzata Gil Jeffrey L. Salisbury Mathew P. Goetz Vera Suman Amy Degnim James McCubrey Tufia Haddad Ianko Iankov Chenye B. Kurokawa Nicole Shumacher James N. Ingle Evanthia Galanis Antonino B. D’Assoro

Although the majority of breast cancers initially respond to the cytotoxic effects of chemotherapeutic agents, most breast cancer patients experience tumor relapse and ultimately die because of drug resistance. Breast cancer cells undergoing epithelial to mesenchymal transition (EMT) acquire a CD44+/CD24-/ALDH1+ cancer stem cell-like phenotype characterized by an increased capacity for tumor se...

Journal: :Molecular cancer therapeutics 2014
Jessica J Huck Mengkun Zhang Jerome Mettetal Arijit Chakravarty Karthik Venkatakrishnan Xiaofei Zhou Rob Kleinfield Marc L Hyer Karuppiah Kannan Vaishali Shinde Andy Dorner Mark G Manfredi Wen Chyi Shyu Jeffrey A Ecsedy

Aurora A kinase orchestrates multiple key activities, allowing cells to transit successfully into and through mitosis. MLN8237 (alisertib) is a selective Aurora A inhibitor that is being evaluated as an anticancer agent in multiple solid tumors and heme-lymphatic malignancies. The antitumor activity of MLN8237 when combined with docetaxel or paclitaxel was evaluated in in vivo models of triple-...

2013
ALEXEY A. LEONTOVICH JEFFREY L. SALISBURY MASSIMILIANO VEROUX TIZIANO TALLARITA DANIEL BILLADEAU JAMES McCUBREY JAMES INGLE EVANTHIA GALANIS ANTONINO B. D’ASSORO

Centrosome amplification plays a key role in the origin of chromosomal instability (CIN) during cancer development and progression. In this study, MCF-7 breast cancer cell lines harboring abrogated p53 function (vMCF-7DNp53) were employed to investigate the relationship between induction of genotoxic stress, activation of cyclin-A/Cdk2 and Aurora-A oncogenic signalings and development of centro...

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