نتایج جستجو برای: chlorotoxin like peptide

تعداد نتایج: 792662  

Journal: :Journal of medicinal chemistry 2015
Huy N Hoang Kun Song Timothy A Hill David R Derksen David J Edmonds W Mei Kok Chris Limberakis Spiros Liras Paula M Loria Vincent Mascitti Alan M Mathiowetz Justin M Mitchell David W Piotrowski David A Price Robert V Stanton Jacky Y Suen Jane M Withka David A Griffith David P Fairlie

Cyclic constraints are incorporated into an 11-residue analogue of the N-terminus of glucagon-like peptide-1 (GLP-1) to investigate effects of structure on agonist activity. Cyclization through linking side chains of residues 2 and 5 or 5 and 9 produced agonists at nM concentrations in a cAMP assay. 2D NMR and CD spectra revealed an N-terminal β-turn and a C-terminal helix that differentially i...

Journal: :American journal of physiology. Regulatory, integrative and comparative physiology 2002
Linda Rinaman Elizabeth E Rothe

The present study examined possible interactions between central glucagon-like peptide-1 (GLP-1) and oxytocin (OT) neural systems by determining whether blockade of GLP-1 receptors attenuates OT-induced anorexia and vice versa. Male rats were acclimated to daily 4-h food access. In the first experiment, rats were infused centrally with GLP-1 receptor antagonist or vehicle, followed by an anorex...

2013
Hitoshi Ando Kentarou Ushijima Akio Fujimura

Circadian clocks in peripheral tissues are powerfully entrained by feeding. The mechanisms underlying this food entrainment remain unclear, although various humoral and neural factors have been reported to affect peripheral clocks. Because glucagon-like peptide-1 (GLP-1), which is rapidly secreted in response to food ingestion, influences multiple humoral and neural signaling pathways, we sugge...

Journal: :Comparative biochemistry and physiology. Part B, Biochemistry & molecular biology 2001
J T Silverstein V M Bondareva J B Leonard E M Plisetskaya

Glucagon-like peptide 1 is a compound known to cause reduced food intake in mammals, though its action on feed intake in fish is unknown. The clear differences in the effects of GLP-1 on mammalian and teleostean glucose homeostasis suggest that we cannot assume a similar action of GLP-1 on feeding in mammals and fish. In this study the effects and specificity of centrally administered GLP-1 on ...

Journal: :American journal of physiology. Gastrointestinal and liver physiology 2013
Yuji Nakamura Takanori Kanai Keita Saeki Miho Takabe Junichiro Irie Jun Miyoshi Yohei Mikami Toshiaki Teratani Takahiro Suzuki Naoteru Miyata Tadakazu Hisamatsu Nobuhiro Nakamoto Yoshiyuki Yamagishi Hajime Higuchi Hirotoshi Ebinuma Shigenari Hozawa Hidetsugu Saito Hiroshi Itoh Toshifumi Hibi

Glucagon-like peptide-1 (GLP-1) promotes insulin release; however, the relationship between the GLP-1 signal and chronic pancreatitis is not well understood. Here we focus on chemokine (C-C motif) ligand 2 (CCL2) and its receptor (CCR2) axis, which regulates various immune cells, including macrophages, to clarify the mechanism of GLP-1-mediated insulin secretion in chronic pancreatitis in mice....

2016
Yuichiro Yamada Katsushi Tsukiyama Takehiro Sato Tatsunori Shimizu Hiroki Fujita Takuma Narita

The hormonal factors implicated as transmitters of signals from the gut to pancreatic β-cells are referred to as incretins. Gastric inhibitory polypeptide (GIP) and glucagon-like peptide-1 (GLP-1) are incretins. In addition to the insulinotropic effects, we have shown, using the GIP receptor and GLP-1 receptor-deficient mice, that GIP and GLP-1 have direct actions on adipocytes and the kidney, ...

2013
Katsunori Nonogaki Marina Suzuki

Glucagon-like peptide-1 (GLP-1), an insulinotropic gastrointestinal peptide that is primarily produced by intestinal endocrine L-cells, stimulates satiety. Ghrelin, a hormone that is produced predominantly by the stomach stimulates hunger. There are two forms of ghrelin: active ghrelin and inactive des-acyl ghrelin. After depriving mice of food for 24 h, we demonstrated that the systemic admini...

2013
Stefan Trapp James E Richards

Glucagon-like peptide-1 (GLP-1) is both a peripherally expressed incretin and a centrally active neuropeptide. Brain derived GLP-1, produced in preproglucagon (PPG) neurons located in the nucleus of the solitary tract (NTS) and projecting to numerous brain regions, is ideally placed to activate central GLP-1 receptors in a range of autonomic control areas. In vivo analysis of central GLP-1 usin...

Journal: :Journal of the Turkish Chemical Society, Section A: Chemistry 2018

نمودار تعداد نتایج جستجو در هر سال

با کلیک روی نمودار نتایج را به سال انتشار فیلتر کنید