نتایج جستجو برای: antimalarial agents

تعداد نتایج: 366169  

2016
Mithun Rudrapal Dipak Chetia

Malaria disease continues to be a major health problem worldwide due to the emergence of multidrug-resistant strains of Plasmodium falciparum. In recent days, artemisinin (ART)-based drugs and combination therapies remain the drugs of choice for resistant P. falciparum malaria. However, resistance to ART-based drugs has begun to appear in some parts of the world. Endoperoxide compounds (natural...

Journal: :Journal of Enzyme Inhibition and Medicinal Chemistry 2017

اسدالهی, اقباله, اونیل, پروفسور پال, خسروی, افرا,

Background and Objective: Resistance to chloroquine (CQ) in Plasmodium falciparum malaria has become a major health concern in the developing countries. This problem has prompted investigators for finding alternative antimalarials that may be effective against resistant strains. Amodiaquine (AQ) is an antimalarial which is effective against many chloroquine-resistant strains of P. falciparum. H...

Journal: :The American journal of tropical medicine and hygiene 2004
Clinton K Murray Michael W Ellis Duane R Hospenthal

Leptospirosis has recently been described to cause concomitant infection with malaria. Only doxycycline has proven to have chemoprophylactic and therapeutic efficacy for both malaria and leptospirosis. To assess whether other traditional antimalarial agents have antileptospiral activity, we performed broth microdilution susceptibility testing of 16 Leptospira serovars (6 species/14 serogroups) ...

2016
Dipak Chetia Mithun Rudrapal

In this article, a review on bioactive flavonoids that are abundant in medicinal and functional food (dietary) plants has been made, with special reference to antimalarial flavonoid molecules. Flavonoids have been found to exist in plants/plant medicines with a wide structural diversity consisting of numerous polyphenolic compounds and having well defined molecular target specificity. These phy...

Journal: :Journal of chemical information and modeling 2013
Liying Zhang Denis Fourches Alexander Sedykh Hao Zhu Alexander Golbraikh Sean Ekins Julie Clark Michele C. Connelly Martina Sigal Dena Hodges Armand Guiguemde R. Kiplin Guy Alexander Tropsha

Quantitative structure-activity relationship (QSAR) models have been developed for a data set of 3133 compounds defined as either active or inactive against P. falciparum. Because the data set was strongly biased toward inactive compounds, different sampling approaches were employed to balance the ratio of actives versus inactives, and models were rigorously validated using both internal and ex...

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