نتایج جستجو برای: neuropathy target esterase

تعداد نتایج: 449439  

Journal: :Bioorganic & medicinal chemistry letters 2003
Yoffi Segall Gary B Quistad Daniel K Nomura John E Casida

Arachidonylsulfonyl fluoride (3), reported here for the first time, is similar in potency to its known methyl arachidonylfluorophosphonate (2) analogue as an inhibitor of mouse brain fatty acid amide hydrolase activity (IC(50) 0.1 nM) and cannabinoid CB1 agonist [3H]CP 55,940 binding (IC(50) 304-530 nM). Interestingly, 3 is much more selective than 2 as an inhibitor for fatty acid amide hydrola...

Journal: :Nature communications 2015
S Kmoch J Majewski V Ramamurthy S Cao S Fahiminiya H Ren I M MacDonald I Lopez V Sun V Keser A Khan V Stránecký H Hartmannová A Přistoupilová K Hodaňová L Piherová L Kuchař A Baxová R Chen O G P Barsottini A Pyle H Griffin M Splitt J Sallum J L Tolmie J R Sampson P Chinnery E Banin D Sharon S Dutta R Grebler C Helfrich-Foerster J L Pedroso D Kretzschmar M Cayouette R K Koenekoop

Blindness due to retinal degeneration affects millions of people worldwide, but many disease-causing mutations remain unknown. PNPLA6 encodes the patatin-like phospholipase domain containing protein 6, also known as neuropathy target esterase (NTE), which is the target of toxic organophosphates that induce human paralysis due to severe axonopathy of large neurons. Mutations in PNPLA6 also cause...

Journal: :The Journal of neuroscience : the official journal of the Society for Neuroscience 2005
Max Mühlig-Versen Alexandre Bettencourt da Cruz Jakob-Andreas Tschäpe Markus Moser Reinhard Büttner Karin Athenstaedt Paul Glynn Doris Kretzschmar

The Drosophila Swiss cheese (sws) mutant is characterized by progressive degeneration of the adult nervous system, glial hyperwrapping, and neuronal apoptosis. The Swiss cheese protein (SWS) shares 39% sequence identity with human neuropathy target esterase (NTE), and a brain-specific deletion of SWS/NTE in mice causes a similar pattern of progressive neuronal degeneration. NTE reacts with orga...

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