نتایج جستجو برای: imidazolide

تعداد نتایج: 66  

Journal: :The journal of physical chemistry. A 2007
Stephanie M Villano Adam J Gianola Nicole Eyet Takatoshi Ichino Shuji Kato Veronica M Bierbaum W Carl Lineberger

The 351.1 nm photoelectron spectra of the N-methyl-5-pyrazolide anion and the N-methyl-5-imidazolide anion are reported. The photoelectron spectra of both isomers display extended vibrational progressions in the X2A' ground states of the corresponding radicals that are well reproduced by Franck-Condon simulations, based on the results of B3LYP/6-311++G(d,p) calculations. The electron affinities...

Journal: :The Journal of pharmacology and experimental therapeutics 2010
Lauren M Aleksunes Michael J Goedken Cheryl E Rockwell Juergen Thomale Jose E Manautou Curtis D Klaassen

The use of the chemotherapeutic drug cisplatin is limited in part by nephrotoxicity. Cisplatin causes renal DNA adducts and oxidative stress in rodents. The transcription factor Nrf2 (nuclear factor E2-related factor 2) induces expression of cytoprotective genes, including Nqo1 (NADPH:quinone oxidoreductase 1), Ho-1 (heme oxygenase-1), and Gclc (glutamate cysteine ligase catalytic subunit), in ...

Journal: :Molecular cancer therapeutics 2007
Melinda S Yates Masafumi Tauchi Fumiki Katsuoka Kathleen C Flanders Karen T Liby Tadashi Honda Gordon W Gribble Delinda A Johnson Jeffrey A Johnson Neal C Burton Tomás R Guilarte Masayuki Yamamoto Michael B Sporn Thomas W Kensler

Synthetic triterpenoids have been developed, which are potent inducers of cytoprotective enzymes and inhibitors of inflammation, greatly improving on the weak activity of naturally occurring triterpenoids. An imidazolide triterpenoid derivative, 1-[2-cyano-3,12-dioxooleana-1,9(11)-dien-28-oyl]imidazole (CDDO-Im or TP235), has been previously shown to potently protect against hepatic tumorigenes...

Journal: :Cancer research 2005
Karen Liby Thomas Hock Mark M Yore Nanjoo Suh Andrew E Place Renee Risingsong Charlotte R Williams Darlene B Royce Tadashi Honda Yukiko Honda Gordon W Gribble Nathalie Hill-Kapturczak Anupam Agarwal Michael B Sporn

The synthetic triterpenoid 2-cyano-3,12-dioxooleana-1,9(11)-dien-28-oic acid (CDDO) and its derivative 1-[2-cyano-3-,12-dioxooleana-1,9(11)-dien-28-oyl]imidazole (CDDO-Im) are multifunctional molecules with potent antiproliferative, differentiating, and anti-inflammatory activities. At nanomolar concentrations, these agents rapidly increase the expression of the cytoprotective heme oxygenase-1 ...

2017
Dongwei Xu Lili Chen Xiaosong Chen Yankai Wen Chang Yu Jufang Yao Hailong Wu Xin Wang Qiang Xia Xiaoni Kong

Nuclear factor erythroid 2-related factor 2 (Nrf2)-mediated induction of antioxidants has been implicated to have protective roles in ischemia-reperfusion (I/R) injury in many animal models. However, the in vivo effects of CDDO-imidazole (CDDO-Im) (1-[2-cyano-3-,12-dioxooleana-1,9(11)-dien-28-oyl] imidazole), a Nrf2 activator, in hepatic I/R injury is lacking and its exact molecular mechanisms ...

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