نتایج جستجو برای: telaprevir

تعداد نتایج: 686  

2010

Telaprevir (LY 570310; LY-570310; LY570310; MP 424; MP-424; VX 950; VX-950) is an orally administered peptidomimetic inhibitor of the hepatitis C virus (HCV) protease NS3/4A. It is being developed by Vertex Pharmaceuticals and its licensees for the treatment of HCV infections and has recently been submitted to the US FDA for approval. As the first ever HCV protease inhibitor in phase III develo...

Journal: :ACS chemical biology 2015
Jean Ndjomou M Josie Corby Noreena L Sweeney Alicia M Hanson Cihan Aydin Akbar Ali Celia A Schiffer Kelin Li Kevin J Frankowski Frank J Schoenen David N Frick

This study examines the specificity and mechanism of action of a recently reported hepatitis C virus (HCV) nonstructural protein 3 (NS3) helicase-protease inhibitor (HPI), and the interaction of HPI with the NS3 protease inhibitors telaprevir, boceprevir, danoprevir, and grazoprevir. HPI most effectively reduced cellular levels of subgenomic genotype 4a replicons, followed by genotypes 3a and 1...

Journal: :Hawai'i journal of medicine & public health : a journal of Asia Pacific Medicine & Public Health 2013
Matthew J Akiyama Joy I Piotrowski Marina M Roytman Siu M A Chan Leena K Hong Leslie Huddleston Ruby Trujillo Naoky C S Tsai

Recent advances in treatment of chronic hepatitis C virus have improved significantly due to the introduction of two new protease inhibitors-telaprevir and boceprevir. In combination with the previous standard of care, peginterferon and ribavirin, telaprevir and boceprevir have demonstrated improved sustained virologic response rates for HCV genotype 1 patients by approximately 30%. The purpose...

Journal: :Journal of managed care & specialty pharmacy 2015
T Kim Le Anupama Kalsekar Dendy Macaulay Yong Yuan Rachael A Sorg Christopher R Behrer Jin Wei Eric Q Wu

BACKGROUND Chronic hepatitis C (CHC) is associated with substantial morbidity and mortality, with the future burden of disease predicted to significantly increase. The recent addition of 2 direct-acting antiviral (DAA) protease inhibitors, telaprevir and boceprevir, to peginterferon alfa (PEG) and ribavirin (RBV) therapy has been shown to significantly improve sustained virologic response rates...

2015
Suheyla Komur Behice Kurtaran Ayse Seza Inal Husnu Pullukcu Aslihan Ulu Ferit Kuscu Tansu Yamazhan Yesim Tasova Hasan Salih Zeki Aksu

BACKGROUND In patients with chronic hepatitis C, triple drug regimens containing a protease inhibitor, peginterferon and ribavirin were found to significantly increase sustained virologic response rates compared to dual drug regimen containing pegylated interferon and ribavirin, especially in genotype 1. OBJECTIVES In Turkey, telaprevir has been used since March 2013. We aimed to evaluate res...

Journal: :The Netherlands journal of medicine 2013
M H Lamers M M T J Broekman C A Boucher J T Brouwer D M Burger B van Hoek A I M Hoepelman R J de Knegt H W Reesink J P H Drenth

In this new Dutch guideline for hepatitis C virus infection we provide recommendations for the management of hepatitis C infection. Until 2012 the standard for treatment consisted of pegylated interferon alpha (peg-IFNa) and ribavirin. The advent of first-generation direct antiviral agents such as boceprevir and telaprevir has changed the concept of treatment of adult chronic hepatitis C genoty...

Journal: :Clinical gastroenterology and hepatology : the official clinical practice journal of the American Gastroenterological Association 2013
Kee Chan Mai Ngan Lai Erik J Groessl Amresh D Hanchate John B Wong Jack A Clark Steven M Asch Allen L Gifford Samuel B Ho

BACKGROUND & AIMS The Veterans Health Administration (VHA) is the largest single provider of care for hepatitis C virus (HCV) infection in the United States. We analyzed the cost effectiveness of treatment with the HCV protease inhibitors boceprevir and telaprevir in a defined managed care population of 102,851 patients with untreated chronic genotype 1 infection. METHODS We used a decision-a...

Journal: :Clinical infectious diseases : an official publication of the Infectious Diseases Society of America 2013
Andrea Calcagno Lucio Boglione Francesco Giuseppe De Rosa Giovanni Di Perri Stefano Bonora

BACKGROUND The licensing of direct-acting antivirals heralds a new era in the treatment of hepatitis C virus (HCV) genotype 1. We undertook a mixed treatment comparison to examine the relative efficacy among current treatments for HCV. METHODS A systematic literature review identified relevant studies. Meta-analyses were planned in treatment-naive and treatment-experienced patients. Study arm...

2017
Helena HL Borba Astrid Wiens Laiza M Steimbach Fernanda S Tonin Maria LA Pedroso Cláudia AP Ivantes Fernando Fernandez-Llimos Roberto Pontarolo

BACKGROUND Chronic hepatitis C is a major public health issue, but there is a gap in the literature regarding the effectiveness and safety of direct-acting antiviral agents in the Brazilian population. The main aim of this study was to describe the effectiveness of boceprevir and telaprevir in patients treated at public health care institutions in Brazil. MATERIALS AND METHODS A prospective l...

Journal: :The New England journal of medicine 2011
Stefan Zeuzem Pietro Andreone Stanislas Pol Eric Lawitz Moises Diago Stuart Roberts Roberto Focaccia Zobair Younossi Graham R Foster Andrzej Horban Peter Ferenci Frederik Nevens Beat Müllhaupt Paul Pockros Ruben Terg Daniel Shouval Bart van Hoek Ola Weiland Rolf Van Heeswijk Sandra De Meyer Don Luo Griet Boogaerts Ramon Polo Gaston Picchio Maria Beumont

BACKGROUND Up to 60% of patients with hepatitis C virus (HCV) genotype 1 infection do not have a sustained virologic response to therapy with peginterferon alfa plus ribavirin. METHODS In this randomized, phase 3 trial, we evaluated the addition of telaprevir to peginterferon alfa-2a plus ribavirin in patients with HCV genotype 1 infection who had no response or a partial response to previous...

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