نتایج جستجو برای: jwh133

تعداد نتایج: 38  

2017
Eva Martínez-Pinilla Katia Varani Irene Reyes-Resina Edgar Angelats Fabrizio Vincenzi Carlos Ferreiro-Vera Julen Oyarzabal Enric I. Canela José L. Lanciego Xavier Nadal Gemma Navarro Pier Andrea Borea Rafael Franco

The mechanism of action of cannabidiol (CBD), the main non-psychotropic component of Cannabis sativa L., is not completely understood. First assumed that the compound was acting via cannabinoid CB2 receptors (CB2Rs) it is now suggested that it interacts with non-cannabinoid G-protein-coupled receptors (GPCRs); however, CBD does not bind with high affinity to the orthosteric site of any GPCR. To...

2013
Claudia Compagnucci Sara Di Siena Maria Blaire Bustamante Daniele Di Giacomo Monia Di Tommaso Mauro Maccarrone Paola Grimaldi Claudio Sette

Neural stem cells (NSCs) are self-renewing cells that can differentiate into multiple neural lineages and repopulate regions of the brain after injury. We have investigated the role of endocannabinoids (eCBs), endogenous cues that modulate neuronal functions including neurogenesis, and their receptors CB(1) and CB(2) in mouse NSCs. Real-time PCR and Western blot analyses indicated that CB(1) is...

Journal: :Journal of biomolecular screening 2010
Paola Scandroglio Rossella Brusa Gianluca Lozza Isabella Mancini Roberta Petrò Angelo Reggiani Massimiliano Beltramo

Recently, new technologies based on biosensors and called label free have been developed. These technologies eliminate the need for using markers and dyes. The authors applied one of these technologies, based on measurement of cell impedance variation, to study the pharmacological profiles of ligands for the cannabinoid receptor 2 (CB2), a Gi-coupled receptor, and for the metabopotropic glutama...

Journal: :Glia 2009
Susana Mato Elena Alberdi Catherine Ledent Masahiko Watanabe Carlos Matute

Regulation of Ca(2+) homeostasis plays a critical role in oligodendrocyte function and survival. Cannabinoid CB(1) and CB(2) receptors have been shown to regulate Ca(2+) levels and/or K(+) currents in a variety of cell types. In this study we investigated the effect of cannabinoid compounds on the Ca(2+) influx elicited in cultured oligodendrocytes by transient membrane depolarization with an e...

Journal: :Neuropharmacology 2016
Attila Köfalvi Cristina Lemos Ana M. Martín-Moreno Bárbara S. Pinheiro Luis García-García Miguel A. Pozo Ângela Valério-Fernandes Rui O. Beleza Paula Agostinho Ricardo J. Rodrigues Susana J. Pasquaré Rodrigo A. Cunha María L. de Ceballos

Cannabinoid CB2 receptors (CB2Rs) are emerging as important therapeutic targets in brain disorders that typically involve neurometabolic alterations. We here addressed the possible role of CB2Rs in the regulation of glucose uptake in the mouse brain. To that aim, we have undertaken 1) measurement of (3)H-deoxyglucose uptake in cultured cortical astrocytes and neurons and in acute hippocampal sl...

Journal: :Stroke 2017
Isabel Bravo-Ferrer María I Cuartero Juan G Zarruk Jesús M Pradillo Olivia Hurtado Víctor G Romera Javier Díaz-Alonso Juan M García-Segura Manuel Guzmán Ignacio Lizasoain Ismael Galve-Roperh María A Moro

BACKGROUND AND PURPOSE Stroke is a leading cause of adult disability characterized by physical, cognitive, and emotional disturbances. Unfortunately, pharmacological options are scarce. The cannabinoid type-2 receptor (CB2R) is neuroprotective in acute experimental stroke by anti-inflammatory mechanisms. However, its role in chronic stroke is still unknown. METHODS Stroke was induced by perma...

2002
RENE ANIKWUE JOHN W. HUFFMAN ZACHARY L. MARTIN SANDRA P. WELCH

Cannabinoids have been shown to increase the release of arachadonic acid, whereas nonsteroidal anti-inflammatory drugs (NSAIDs) have been shown to decrease the analgesic effects of cannabinoids. We evaluated the antinociceptive effects of chronic administration of -tetrahydrocannabinol ( -THC), anandamide (an endogenous cannabinoid), arachadonic acid, ethanolamine, and methanandamide on several...

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