نتایج جستجو برای: benserazide

تعداد نتایج: 137  

2015
Michael S. Boosalis Jose I. Sangerman Gary L. White Roman F. Wolf Ling Shen Yan Dai Emily White Levi H. Makala Biaoru Li Betty S. Pace Mehdi Nouraie Douglas V. Faller Susan P. Perrine Andrew C. Wilber

High-level fetal (γ) globin expression ameliorates clinical severity of the beta (β) hemoglobinopathies, and safe, orally-bioavailable γ-globin inducing agents would benefit many patients. We adapted a LCR-γ-globin promoter-GFP reporter assay to a high-throughput robotic system to evaluate five diverse chemical libraries for this activity. Multiple structurally- and functionally-diverse compoun...

2014
Marty Hinz Alvin Stein Ted Cole

The only indication for carbidopa and benserazide is the management of L-3,4-dihydroxyphenylalanine (L-dopa)-induced nausea. Both drugs irreversibly bind to and permanently deactivate pyridoxal 5'-phosphate (PLP), the active form of vitamin B6, and PLP-dependent enzymes. PLP is required for the function of over 300 enzymes and proteins. Virtually every major system in the body is impacted direc...

2014
Cheng-long Xie Wen-Wen Wang Su-fang Zhang Ming-Lu Yuan Jun-Yi Che Jing Gan Lu Song Wei-En Yuan Zhen-Guo Liu

L-3, 4-dihydroxyphenylalanine (L-dopa) is the gold standard for symptomatic treatment of Parkinson's disease (PD), but long-term therapy is associated with the emergence of L-dopa-induced dyskinesia (LID). In the present study, L-dopa and benserazide were loaded by poly (lactic-co-glycolic acid) microspheres (LBM), which can release levodopa and benserazide in a sustained manner in order to con...

2015
Jessica L Kelts James J Cali Sarah J Duellman John Shultz

Induction of oxidative stress by drugs and other xenobiotics is an important mechanism of cytotoxicity. However, in vitro studies on the relationship between oxidative stress and cytotoxicity in cultured cells is frequently complicated by the fact that cell culture medium components affect reactive oxygen species (ROS) exposures in ways that vary with the mode of ROS production. The objectives ...

Journal: :Journal of neurology, neurosurgery, and psychiatry 1988
R J Hardie A J Lees

Twenty six consecutive patients with neuroleptic-induced Parkinson's syndrome (NIPS) are described. Their median age was 61 years, 60% were female, and most had received chronic neuroleptic medication for psychiatric indications. The clinical features were indistinguishable from idiopathic Parkinson's disease, except for the presence of co-existing orofacial chorea, limb dyskinesia or akathisia...

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