نتایج جستجو برای: 17β hydroxysteroid dehydrogenase type1

تعداد نتایج: 75368  

2017
Roger T Engeli Simona R Rohrer Anna Vuorinen Sonja Herdlinger Teresa Kaserer Susanne Leugger Daniela Schuster Alex Odermatt

Parabens are effective preservatives widely used in cosmetic products and processed food, with high human exposure. Recent evidence suggests that parabens exert estrogenic effects. This work investigated the potential interference of parabens with the estrogen-activating enzyme 17β-hydroxysteroid dehydrogenase (17β-HSD) 1 and the estrogen-inactivating 17β-HSD2. A ligand-based 17β-HSD2 pharmacop...

Journal: :Journal of the Brazilian Chemical Society 2019

2017
Ildikó Bacsa Rebeka Jójárt János Wölfling Gyula Schneider Bianka Edina Herman Mihály Szécsi Erzsébet Mernyák

Novel 13α-estrone derivatives were synthesized by Sonogashira coupling. Transformations of 2- or 4-iodo regioisomers of 13α-estrone and its 3-methyl ether were carried out under different conditions in a microwave reactor. The 2-iodo isomers were reacted with para-substituted phenylacetylenes using Pd(PPh3)4 as catalyst and CuI as a cocatalyst. Coupling reactions of 4-iodo derivatives could be ...

2014
Tomomi Yoda Keely May McNamara Yasuhiro Miki Mayu Takagi Yoshiaki Rai Yasuyo Ohi Yasuaki Sagara Kentaro Tamaki Hisashi Hirakawa Takanori Ishida Takashi Suzuki Noriaki Ohuchi Hironobu Sasano

Invasive lobular carcinoma (ILC) accounts for approximately 10% of all breast carcinomas and is characterized by higher levels of androgen receptor (AR) compared to invasive ductal carcinoma (IDC). Despite this potentially androgen-responsive environment, the combined importance of AR and androgen metabolism in non-neoplastic lobules and lobular carcinoma remains unknown. Therefore, in this stu...

2016
Xiaoxiao Gao Kaifa Zhang Min Song Xiumei Li Lei Luo Yuan Tian Yunhai Zhang Yunsheng Li Xiaorong Zhang Yinghui Ling Fugui Fang Ya Liu

Nesfatin-1 is an important molecule in the regulation of reproduction. However, its role in the reproductive axis in male animals remains to be understood. Here, we found that nesfatin-1 was mainly distributed in the arcuate nucleus (ARC), paraventricular nucleus (PVN), periventricular nucleus (PeN), and lateral hypothalamic area (LHA) of the hypothalamus; adenohypophysis and Leydig cells in ma...

Journal: :The Journal of clinical endocrinology and metabolism 2014
Hanna Savolainen-Peltonen Veera Vihma Marjut Leidenius Feng Wang Ursula Turpeinen Esa Hämäläinen Matti J Tikkanen Tomi S Mikkola

CONTEXT It has been shown that breast tumor actively produces and metabolizes steroid hormones. However, little is known about the possible mechanisms through which the nonmalignant adipose tissue contributes to steroid hormone metabolism. OBJECTIVE We compared the metabolic pathways producing active estradiol in breast sc adipose tissue of postmenopausal women with or without breast cancer. ...

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