نتایج جستجو برای: روش rtk

تعداد نتایج: 371594  

Journal: :Science signaling 2013
Joel P Wagner Alejandro Wolf-Yadlin Mark Sevecka Jennifer K Grenier David E Root Douglas A Lauffenburger Gavin MacBeath

Although many anticancer drugs that target receptor tyrosine kinases (RTKs) provide clinical benefit, their long-term use is limited by resistance that is often attributed to increased abundance or activation of another RTK that compensates for the inhibited receptor. To uncover common and unique features in the signaling networks of RTKs, we measured time-dependent signaling in six isogenic ce...

2014
Alexey Goltsov Yusuf Deeni Hilal S. Khalil Tero Soininen Stylianos Kyriakidis Huizhong Hu Simon P. Langdon David J. Harrison James Bown

The receptor tyrosine kinases (RTKs) are key drivers of cancer progression and targets for drug therapy. A major challenge in anti-RTK treatment is the dependence of drug effectiveness on co-expression of multiple RTKs which defines resistance to single drug therapy. Reprogramming of the RTK network leading to alteration in RTK co-expression in response to drug intervention is a dynamic mechani...

Journal: :Proceedings of the National Academy of Sciences of the United States of America 2014
Lijoy K Mathew Nicolas Skuli Vera Mucaj Samuel S Lee Pascal O Zinn Pratheesh Sathyan Hongxia Z Imtiyaz Zhongfa Zhang Ramana V Davuluri Shilpa Rao Sriram Venneti Priti Lal Justin D Lathia Jeremy N Rich Brian Keith Andy J Minn M Celeste Simon

Glioblastoma multiforme (GBM) and the mesenchymal GBM subtype in particular are highly malignant tumors that frequently exhibit regions of severe hypoxia and necrosis. Because these features correlate with poor prognosis, we investigated microRNAs whose expression might regulate hypoxic GBM cell survival and growth. We determined that the expression of microRNA-218 (miR-218) is decreased signif...

Journal: :Molecular cancer research : MCR 2016
Jaclyn F Hechtman Ahmet Zehir Rona Yaeger Lu Wang Sumit Middha Tao Zheng David M Hyman David Solit Maria E Arcila Laetitia Borsu Jinru Shia Efsevia Vakiani Leonard Saltz Marc Ladanyi

UNLABELLED Targeted therapy for metastatic colorectal carcinoma consists of anti-EGFR therapy for patients with RAS/RAF wild-type tumors. However, the response rate remains low, suggesting the presence of alternative drivers possibly also representing potential therapeutic targets. We investigated receptor tyrosine kinase (RTK) alterations and MAP2K1 (MEK1) mutations in a large cohort of colore...

2016
Frédéric G. Brunet Jean-Nicolas Volff Manfred Schartl

The receptor tyrosine kinase (RTK) gene family, involved primarily in cell growth and differentiation, comprises proteins with a common enzymatic tyrosine kinase intracellular domain adjacent to a transmembrane region. The amino-terminal portion of RTKs is extracellular and made of different domains, the combination of which characterizes each of the 20 RTK subfamilies among mammals. We analyze...

Journal: :Development 2006
Lesley A Jarvis Stephanie J Toering Michael A Simon Mark A Krasnow Rachel K Smith-Bolton

Drosophila Corkscrew protein and its vertebrate ortholog SHP-2 (now known as Ptpn11) positively modulate receptor tyrosine kinase (RTK) signaling during development, but how these tyrosine phosphatases promote tyrosine kinase signaling is not well understood. Sprouty proteins are tyrosine-phosphorylated RTK feedback inhibitors, but their regulation and mechanism of action are also poorly unders...

Journal: :Cancer research 2010
Alexander M Xu Paul H Huang

Cancer cells employ multiple mechanisms to evade tightly regulated cellular processes such as proliferation, apoptosis, and senescence. Systems-wide analyses of tumors have recently identified receptor tyrosine kinase (RTK) coactivation as an important mechanism by which cancer cells achieve chemoresistance. This mini-review discusses our current understanding of the complex and dynamic process...

Journal: :Molecular and cellular biology 2004
Andrea Pomrehn Myers Laura B Corson Janet Rossant Julie C Baker

Receptor tyrosine kinase (RTK) signals regulate the specification of a varied array of tissue types by utilizing distinct modules of proteins to elicit diverse effects. The RSK proteins are part of the RTK signal transduction pathway and are thought to relay these signals by acting downstream of extracellular signal-regulated kinase (ERK). In this study we report the identification of ribosomal...

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