نتایج جستجو برای: polystyrene n alanine sulfonamide

تعداد نتایج: 1011197  

Journal: :Organic & biomolecular chemistry 2018
Yali Zhou Dengke Li Shi Tang Hongwei Sun Jinbo Huang Qiang Zhu

A facile construction of the spiro[indole-3,2'-pyrrolidine] skeleton, through diacetoxyiodobenzene (PIDA) mediated C-N bond-forming dearomatization of C3 sulfonamide linked indole derivatives, has been developed. A variety of spiro-indolepyrrolidines were obtained in moderate to excellent yields under mild conditions.

2014
Stephen Brand Neil R. Norcross Stephen Thompson Justin R. Harrison Victoria C. Smith David A. Robinson Leah S. Torrie Stuart P. McElroy Irene Hallyburton Suzanne Norval Paul Scullion Laste Stojanovski Frederick R. C. Simeons Daan van Aalten Julie A. Frearson Ruth Brenk Alan H. Fairlamb Michael A. J. Ferguson Paul G. Wyatt Ian H. Gilbert Kevin D. Read

Trypanosoma brucei N-myristoyltransferase (TbNMT) is an attractive therapeutic target for the treatment of human African trypanosomiasis (HAT). From previous studies, we identified pyrazole sulfonamide, DDD85646 (1), a potent inhibitor of TbNMT. Although this compound represents an excellent lead, poor central nervous system (CNS) exposure restricts its use to the hemolymphatic form (stage 1) o...

Journal: :Organic Letters 2021

A highly diastereoselective, visible-light-induced [3 + 2] cycloaddition between N-sulfonyl cyclopropylamines and electron-deficient olefins is reported. The reactions proceed via the oxidation of a sulfonamide aza-anion by an organic photocatalyst to generate nitrogen-centered radical. Strain-induced ring opening intermolecular addition olefin intermediate carbon-centered radical that reduced ...

Journal: :Antimicrobial agents and chemotherapy 2003
Désirée E Bennett Mary T Cafferkey

We identified a previously undocumented mutation in the dihydropteroate synthase (folP) gene associated with Neisseria meningitidis sulfonamide resistance. A PCR-based assay to detect this mutation, which is 100% predictive of sulfonamide resistance, was developed.

Journal: :Molecules 2016
Kei Saito Koji Miyamoto Sepa Nanayakkara Hirotaka Ihara Milton T W Hearn

A new solid phase catalyst, poly(N-4-vinylbenzyl-1,4,7-triazacyclononane) copper(I) complex, grafted onto polystyrene particles, has been employed for the oxidative polymerization of 2,6-dimethylphenol using an aqueous biphasic (water/toluene) solvent system. The solid catalyst was synthesized by first grafting N-(4-vinylbenzyl)-1,4,7-triaza-cyclononane onto polystyrene particles using a radica...

Journal: :Soft matter 2014
Xi-Xian Ke Lian Wang Jun-Ting Xu Bin-Yang Du Ying-Feng Tu Zhi-Qiang Fan

The effect of temperature on the micellar morphology of two polystyrene-b-poly(N-isopropylacrylamide) (PS-b-PNIPAM) diblock copolymers in an aqueous solution was investigated by dynamic light scattering (DLS) and transmission electron microscopy (TEM). At 25 °C, a mixture of vesicles and spheres are observed for the micelles of PS65-b-PNIPAM108, while PS65-b-PNIPAM360 exhibits mixed cylindrical...

Journal: :Macromolecular Chemistry and Physics 2022

The synthesis of well-defined homo- and co-polypeptides L-alanine (L-Ala) by ring-opening polymerization (ROP) its N-carboxyanhydride (NCAs), either via suspension/interfacial- or solution phase-polymerization using 10-undecene-1-amine ?,?-diamino poly(ethylene glycol) (8 1.5 kDa) as primary amine initiators is reported. When conducting ROP NCA-alanine under suspension/interfacial conditions, b...

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