نتایج جستجو برای: non ulcerogenic

تعداد نتایج: 1317118  

Journal: :Drug metabolism and pharmacokinetics 2013
Naoki Yamakawa Shintaro Suemasu Hiroshi Watanabe Kayoko Tahara Ken-ichiro Tanaka Yoshinari Okamoto Masami Ohtsuka Toru Maruyama Tohru Mizushima

  We recently reported that, compared to loxoprofen (LOX, an non-steroidal anti-inflammatory drug), the LOX derivative fluoro-loxoprofen (F-LOX) is less ulcerogenic but has similar anti-inflammatory activity. Our previous in vitro studies suggested that both LOX and F-LOX are pro-drugs, the active metabolites of which are their trans-alcohol forms. In this study, we compared the pharmacokinetic...

2017
Ka-Shing Cheung Wai K Leung

Novel oral anticoagulants (NOACs), which include direct thrombin inhibitor (dabigatran) and direct factor Xa inhibitors (rivaroxaban, apixaban and edoxaban), are gaining popularity in the prevention of embolic stroke in non-valvular atrial fibrillation as well as in the prevention and treatment of venous thromboembolism. However, similar to traditional anticoagulants, NOACs have the side effect...

پایان نامه :وزارت علوم، تحقیقات و فناوری - دانشگاه صنعتی شیراز - دانشکده مهندسی برق و الکترونیک 1393

در این پایان نامه با استفاده از تابع لیاپانوف فازی، به طراحی کنترل کننده pdc و non-pdc برای سیستم های فازی افاین پرداخته می شود. استفاده از تابع لیاپانوف فازی باعث برقراری راحت تر شرایط پایداری و در نتیجه کاهش محافظه کاری می شود. همچنین استفاده از این تابع لیاپانوف به منظور پایدارسازی، طیف گسترده تری از سیستم های فازی افاین را شامل می شود. از طرفی استفاده از کنترل کننده non-pdc باعث می شود شرای...

2014
Thais Regina Ferreira de Melo Rafael Consolin Chelucci Maria Elisa Lopes Pires Luiz Antonio Dutra Karina Pereira Barbieri Priscila Longhin Bosquesi Gustavo Henrique Goulart Trossini Man Chin Chung Jean Leandro dos Santos

A series of anti-inflammatory derivatives containing an N-acyl hydrazone subunit (4a-e) were synthesized and characterized. Docking studies were performed that suggest that compounds 4a-e bind to cyclooxygenase (COX)-1 and COX-2 isoforms, but with higher affinity for COX-2. The compounds display similar anti-inflammatory activities in vivo, although compound 4c is the most effective compound fo...

Journal: :Planta medica 2007
Ana Carla Carvalho Marjorie M Guedes Antonia L de Souza Maria T Trevisan Alana F Lima Flávia A Santos Vietla S Rao

In search of novel gastroprotective agents, mangiferin, a naturally occurring glucosylxanthone from Mangifera indica L. (Anacardiaceae), was evaluated in mice on gastric injury induced by ethanol and indomethacin. The effects of mangiferin on gastric mucosal damage were assessed by determination of changes in mean gastric lesion area or ulcer score in mice and on gastric secretory volume and to...

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