نتایج جستجو برای: glucuronosyltransferase

تعداد نتایج: 2005  

Journal: :Drug metabolism and disposition: the biological fate of chemicals 2012
Liping Ma Jianguo Sun Ying Peng Rong Zhang Feng Shao Xiaoling Hu Jianping Zhu Xiaojin Wang Xuefang Cheng Yinci Zhu Ping Wan Dong Feng Hui Wu Guangji Wang

Edaravone was launched in Japan in 2001 and was the first neuroprotectant developed for the treatment of acute cerebral infarction. Edaravone is mainly eliminated as glucuronide conjugate in human urine (approximately 70%), but the mechanism involved in the elimination pathway remains unidentified. We investigated the glucuronidation of edaravone in human liver microsomes (HLM) and human kidney...

Journal: :Toxicology 2009
Julien Leghait Véronique Gayrard Nicole Picard-Hagen Marion Camp Elisabeth Perdu Pierre-Louis Toutain Catherine Viguié

Fipronil is a widely used phytosanitary product and insecticide for pets. In the rat, fipronil can disrupt thyroid function by decreasing plasma concentrations of total thyroxine (T4) likely through increased T4 clearance. However, the mechanism of fipronil action on thyroid function remains unclear. The goals of the present study were to evaluate the effects of fipronil on thyroid hormone (TH)...

Journal: :The Journal of biological chemistry 2003
Philip A Gregory Dione A Gardner-Stephen Rikke H Lewinsky Kym N Duncliffe Peter I Mackenzie

The human UDP-glucuronosyltransferases, UGT1A8, 1A9, and 1A10, are closely related in sequence and have a major role in the elimination of lipophilic chemicals by glucuronidation. UGT1A8 and 1A10 are expressed exclusively in the gastrointestinal tract, whereas UGT1A9 is expressed mainly in the liver and kidneys. To determine the factors contributing to the extrahepatic expression of these UDP-g...

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