نتایج جستجو برای: ara h 2

تعداد نتایج: 2822627  

Journal: :Blood 1989
V Gandhi B Nowak M J Keating W Plunkett

Our previous studies indicated that K562 cells loaded with arabinosyl-2-fluoroadenine 5'-triphosphate (F-ara-ATP) accumulated arabinosylcytosine 5'-triphosphate (ara-CTP) at a threefold higher rate compared to the control cells. In the present study lymphocytes were obtained from patients with chronic lymphocytic leukemia before and after F-ara-A monophosphate therapy. The rate of ara-CTP accum...

Journal: :Journal of clinical oncology : official journal of the American Society of Clinical Oncology 2012
Stefan Faderl Meir Wetzler David Rizzieri Gary Schiller Madan Jagasia Robert Stuart Siddhartha Ganguly David Avigan Michael Craig Robert Collins Michael Maris Tibor Kovacsovics Stuart Goldberg Karen Seiter Parameswaran Hari Jochen Greiner Norbert Vey Christian Recher Farhad Ravandi Eunice S Wang Michael Vasconcelles Dirk Huebner Hagop M Kantarjian

PURPOSE To compare the receipt of clofarabine plus cytarabine (Clo+Ara-C arm) with cytarabine (Ara-C arm) in patients ≥ 55 years old with refractory or relapsed acute myelogenous leukemia (AML). PATIENTS AND METHODS Patients were randomly assigned to receive either clofarabine (Clo) 40 mg/m(2) or a placebo followed by Ara-C 1 g/m(2) for five consecutive days. The primary end point was overall...

Journal: :European journal of pharmacology 1998
S Ben-Shabat E Fride T Sheskin T Tamiri M H Rhee Z Vogel T Bisogno L De Petrocellis V Di Marzo R Mechoulam

2-Arachidonoyl-glycerol (2-Ara-GI) has been isolated from various tissues and identified as an endogenous ligand for both cannabinoid receptors, CB1 and CB2. Here we report that in spleen, as in brain and gut, 2-Ara-GI is accompanied by several 2-acyl-glycerol esters, two major ones being 2-linoleoyl-glycerol (2-Lino-Gl) and 2-palmitoyl-glycerol (2-Palm-Gl). These two esters do not bind to the ...

Journal: :Clinical and Translational Allergy 2014

Journal: :Antimicrobial agents and chemotherapy 1991
P de Miranda T C Burnette K K Biron R L Miller D R Averett T A Krenitsky

6-Methoxypurine arabinoside (ara-M) exhibits potent activity against varicella-zoster virus (VZV) as a result of ara-M's anabolism to the triphosphate of adenine arabinoside (ara-ATP) in VZV-infected cells. The adenosine deaminase inhibitor erythro-9-(2-hydroxy-3-nonyl)adenine (EHNA) enhanced the formation of ara-ATP by inhibiting ara-M demethoxylation. In contrast, deoxycoformycin and coformyc...

Journal: :The Journal of clinical investigation 1978
K J Champney C B Lauter E J Bailey A M Lerner

The minimum inhibitory concentration (MIC) of adenine arabinoside (ara-A) in rabbit kidney microtiter tissue cultures (RK-13) to a prototype strain of herpes simplex virus, type 1 (E115) based upon inhibition of cytopathic effects is 1.5 mug/ml. In this system, the MIC of arabinosylhypoxanthine (ara-Hx), the major in vivo metabolic derivative of ara-A, is 75 mug/ml. Inhibition of cytopathic eff...

Journal: :Organic & biomolecular chemistry 2009
Nao Hirata Yusuke Fujisawa Kazuhito Tanabe Hiroshi Harada Masahiro Hiraoka Sei-ichi Nishimoto

An anti-tumour agent of cytarabine (ara-C) was conjugated with a 2-oxopropyl group at the N(4) position to obtain a radiation-activated prodrug (oxo-ara-C) that targeted hypoxic tumour tissues with selective cytotoxicity. The parent anti-tumour agent, ara-C, was confirmed to be released from oxo-ara-Cvia one-electron reduction upon hypoxic X-ray treatment. The prodrug oxo-ara-C had dramatically...

Journal: :Clinical and Translational Allergy 2014

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