نتایج جستجو برای: vasicinone

تعداد نتایج: 24  

Journal: :Zeitschrift fur Naturforschung. C, Journal of biosciences 2014
Mohamed A El-Shanawany Hanaa M Sayed Sabrin R M Ibrahim Marwa A A Fayed

Re-investigation of the methanolic extract of Anisotes trisulcus (Forssk.) Nees aerial parts led to the isolation of two new tricyclic quinazoline alkaloids, 8-amino-7,8,9,11-tetrahydro-6H-pyrido[2,1-b]-quinazoline-2,6-diol (4) and 8-amino-3,6-dihydroxy-7,8,9-trihydro-6H-pyrido[2,1-b]quinazoline-11-one (5), and two quaternary ammonium compounds, (dimethylamino)-N-(hydroxymethyl)-N,N-dimethyl me...

2010
Burkhon Zh. Elmuradov Rasul Ya. Okmanov Asqar Sh. Abdurazakov Bakhodir Tashkhodjaev Khusnutdin M. Shakhidoyatov

The title compound, C(20)H(19)N(3)O, was obtained by condensation of 2,3-dihydro-1H,9H-pyrrolo-[2,1-b]quinazolin-9-one (alkaloid de-oxy-vasicinone, isolated from Peganum Harmala) with 4-(dimethyl-amino)-benzaldehyde in the presence of sodium methoxide. The 2,3-dihydro-1H,9H-pyrrolo-[2,1-b]quinazolin-9-one part of the mol-ecule is roughly planar (r.m.s. deviation = 0.0178 Å) and is essentially c...

2010
P. Nilani B. Duraisamy P. Dhamodaran S. Ravichandran K. Elango

Most exacerbations of asthma can be proven to be associated with bacterial infections and there is scientific evidence that frequent respiratory infections particularly bacterial infections provoke asthma attack. Considering these facts different plant extracts and phytoconstituents with proven anti asthmatic property had been selected for screening anti microbial activity in in-vitro models. I...

2015
Wei Liu Xiaoyuan Shi Yadi Yang Xuemei Cheng Qing Liu Han Han Baohua Yang Chunyong He Yongli Wang Bo Jiang Zhengtao Wang Changhong Wang

Vasicine (VAS), a potential natural cholinesterase inhibitor, exhibited promising anticholinesterase activity in preclinical models and has been in development for treatment of Alzheimer's disease. This study systematically investigated the in vitro and in vivo metabolism of VAS in rat using ultra performance liquid chromatography combined with electrospray ionization quadrupole time-of-flight ...

2013
T. Susila Satyanarayana Reddy

Adathoda vasica is a medicinal plant beneficial for the treatment of asthma, cough, haemorragic disorders, hepatitis and fevers. The leaves of the plant contain a mixture of alkaloid i.e., vasicine and vasicinone. Vasicine has numerous pharmacological activities viz., anti-malarial, anti-inflammatory, antioxidant, antidiabetic, anti-bacterial etc. The study on influence of IBA and NAA on rootin...

Journal: :Archives of pharmacal research 2009
Xi-yuan Zheng Zi-jia Zhang Gui-xin Chou Tao Wu Xue-mei Cheng Chang-hong Wang Zheng-tao Wang

Acetylcholinesterase inhibitors (AChEIs) currently form the basis of the newest drugs available for the treatment of Alzheimer's disease. For the aim of screening effective AChEIs, the methanol extracts of the seeds of genus Peganum were found to show significant inhibitory activity of acetylcholinesterase enzyme (AChE) using an in vitro TLC-bioautographic assay. In further studies to seed of P...

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