نتایج جستجو برای: trichostatin a

تعداد نتایج: 13431797  

Journal: :The Journal of biological chemistry 1999
A Verdel S Khochbin

The histone deacetylase domain of almost all members of higher eukaryotic histone deacetylases already identified (HDAC family) is highly homologous to that of yeast RPD3. In this paper we report the cloning of two cDNAs encoding members of a new family of histone deacetylase in mouse that show a better homology to yeast HDA1 histone deacetylase. These cDNAs encode relatively large proteins, pr...

Journal: :The EMBO journal 2003
Oliver H Krämer Ping Zhu Heather P Ostendorff Martin Golebiewski Jens Tiefenbach Marvin A Peters Boris Brill Bernd Groner Ingolf Bach Thorsten Heinzel Martin Göttlicher

Histone-modifying enzymes play essential roles in physiological and aberrant gene regulation. Since histone deacetylases (HDACs) are promising targets of cancer therapy, it is important to understand the mechanisms of HDAC regulation. Selective modulators of HDAC isoenzymes could serve as efficient and well-tolerated drugs. We show that HDAC2 undergoes basal turnover by the ubiquitin-proteasome...

2013
Cheryl V. Rahman Stuart J. Smith Paul S. Morgan Keith A. Langmack Phil A. Clarke Alison A. Ritchie Donald C. Macarthur Felicity R. Rose Kevin M. Shakesheff Richard G. Grundy Ruman Rahman

INTRODUCTION Polymer-based delivery systems offer innovative intra-cavity administration of drugs, with the potential to better target micro-deposits of cancer cells in brain parenchyma beyond the resected cavity. Here we evaluate clinical utility, toxicity and sustained drug release capability of a novel formulation of poly(lactic-co-glycolic acid) (PLGA)/poly(ethylene glycol) (PEG) microparti...

2014
Huang Ying Mao-Chun Xu Jing-Hua Tan Jing-Hua Shen Hao Wang Dai-Fu Zhang

Pressure overload induces cardiac hypertrophy through activation of Janus kinase 2 (Jak2), however, the underlying mechanisms remain largely unknown. In the current study, we tested whether histone deacetylase 2 (HDAC2) was involved in the process. We found that angiotensin II (Ang-II)-induced re-expression of fetal genes (Atrial natriuretic peptide (ANP) and brain natriuretic peptide (BNP)) in...

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