نتایج جستجو برای: platin

تعداد نتایج: 431  

2016
María José Echarri Ana Lopez-Martin Ricardo Hitt

Surgery and radiotherapy are the standard treatment options for patients with squamous cell carcinoma of the head and neck (SCCHN). Chemoradiotherapy is an alternative for patients with locally advanced disease. In recurrent/metastatic disease and after progression to platin-based regimens, no standard treatments other than best supportive care are currently available. Most SCCHN tumours overex...

Journal: :Archives of biochemistry and biophysics 2015
Jie Chen Tian Lan Weimin Zhang Lijia Dong Nan Kang Ming Fu Bing Liu Kangtai Liu Cuixiang Zhang Jincai Hou Qimin Zhan

The clinical efficacy of cisplatin in esophageal squamous cell carcinoma (ESCC) treatment remains undesirable. Src, a non-receptor tyrosine kinase involved in multiple fields of tumorigenesis, recently has been indicated as a promising therapeutic target in the treatment of solid tumors including ESCC. However, whether inhibition of Src activity can increase cisplatin efficacy in ESCC cells rem...

Journal: : 2023

Amaç: Sisplatin, klinikte kanser hastalarının tedavisinde başarılı bir şekilde kullanılmasına rağmen hastalarda rezistans gelişimi ve ciddi toksik yan etkiler görülmektedir. Bu dezavantajların önüne geçmek için bu çalışmada 2,5(6)-disübstitüebenzimidazol türevi taşıyıcı ligandlar kullanarak platin(II) komplekslerinin sentezlenmesi sitotoksik etkilerinin test edilmesi amaçlanmıştır.
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