نتایج جستجو برای: macrocyclic ionophore

تعداد نتایج: 7696  

Journal: :Animal reproduction science 2000
F Jílek R Hüttelová J Petr M Holubová J Rozinek

In vitro matured pig oocytes were activated using a combined treatment of calcium ionophore A 23187 with cycloheximide. The oocytes were exposed to ionophore (10, 25 or 50 microM) for 0.5, 1, 3, 5 or 7 min and then cultured with cycloheximide (0 or 10 microg/ml) for 6 h. Cycloheximide treatment significantly increased the activation rate of oocytes and the percentage of oocytes that were able t...

Journal: :The Journal of biological chemistry 1972
P W Reed H A Lardy

A23187 is a carboxylic acid antibiotic which simultaneously uncouples oxidative phosphorylation and inhibits ATPase of rat liver mitochondria incubated in a magnesium-free medium. The antibiotic acts as a freely mobile carrier to transport calcium and magnesium, but not potassium, from an aqueous medium buffered at pH 7.4 into a bulk organic phase. A23187 causes a progressive release of endogen...

Journal: :Infection and immunity 1983
D M Smith C E Walsh L R Dechatelet M Waite

The effect of the calcium ionophore A23187 on the release and metabolism of [3H]arachidonic acid was examined in normal polymorphonuclear leukocytes and those obtained from patients with chronic granulomatous disease. The ionophore A23187 which stimulates oxidative metabolism in normal polymorphonuclear leukocytes was ineffective in increasing oxidative metabolism (chemiluminescence) in polymor...

Journal: :Journal of the Brazilian Chemical Society 2007

Journal: :Pure and Applied Chemistry 1979

Journal: :Fertility and sterility 2003
Talia Eldar-Geva Baruch Brooks Ehud J Margalioth Edit Zylber-Haran Michael Gal Sherman J Silber

To describe a successful pregnancy and delivery after calcium ionophore oocyte activation in a normozoospermic patient with previous repeated failed fertilization after intracytoplasmic sperm injection (ICSI).Case report. In vitro fertilization unit in a university affiliated medical center.A couple with 5 years of unexplained primary infertility who had repeated failed fertilization after ICSI...

Journal: :Neurochemistry international 2007
A V Kalueff

Gamma-aminobutyric acid (GABA) type A receptors play a key role in brain inhibitory neurotransmission, and are ligand-activated chloride channels blocked by numerous convulsant ligands. Here we summarize data on binding of picrotoxin, tetrazoles, beta-lactams, bicyclophosphates, butyrolactones and neurotoxic pesticides to GABA-A ionophore, and discuss functional and structural overlapping of th...

Journal: :Biochimica et Biophysica Acta (BBA) - Biomembranes 2000

Journal: :Neuron 2008
Paul A. Adlard Robert A. Cherny David I. Finkelstein Elisabeth Gautier Elysia Robb Mikhalina Cortes Irene Volitakis Xiang Liu Jeffrey P. Smith Keyla Perez Katrina Laughton Qiao-Xin Li Susan A. Charman Joseph A. Nicolazzo Simon Wilkins Karolina Deleva Toni Lynch Gaik Kok Craig W. Ritchie Rudolph E. Tanzi Roberto Cappai Colin L. Masters Kevin J. Barnham Ashley I. Bush

As a disease-modifying approach for Alzheimer's disease (AD), clioquinol (CQ) targets beta-amyloid (Abeta) reactions with synaptic Zn and Cu yet promotes metal uptake. Here we characterize the second-generation 8-hydroxy quinoline analog PBT2, which also targets metal-induced aggregation of Abeta, but is more effective as a Zn/Cu ionophore and has greater blood-brain barrier permeability. Given...

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