نتایج جستجو برای: antimycobacterial agents

تعداد نتایج: 361721  

Journal: :ACS chemical biology 2015
Virginia A Kincaid Nir London Kittikhun Wangkanont Darryl A Wesener Sarah A Marcus Annie Héroux Lyudmila Nedyalkova Adel M Talaat Katrina T Forest Brian K Shoichet Laura L Kiessling

Galactofuranose (Galf) is present in glycans critical for the virulence and viability of several pathogenic microbes, including Mycobacterium tuberculosis, yet the monosaccharide is absent from mammalian glycans. Uridine 5'-diphosphate-galactopyranose mutase (UGM) catalyzes the formation of UDP-Galf, which is required to produce Galf-containing glycoconjugates. Inhibitors of UGM have therefore ...

Journal: :Antibiotics 2023

In 2022, we opened an outpatient clinic for the management of polypharmacy and potential drug–drug interactions (pDDIs) in patients with mycobacterial infection (called GAP-MyTB). All who underwent a GAP-MyTB visit from March 2022 to 2023 were included this retrospective analysis. Fifty-two database. They given 10.4 ± 3.7 drugs (2.8 1.0 7.8 3.9 were, respectively, antimycobacterial agents co-me...

2015
Kamaleddin Haj Mohammad Ebrahim Tehrani Vida Mashayekhi Parisa Azerang Somayeh Minaei Soroush Sardari Farzad Kobarfard

A series of cyclic analogues of bioactive thiosemicarbazide derivatives have been synthesized as potential antimycobacterial agents. The 4-amino-1,2,4-triazole-5-thione analogues (Ia-f) were prepared by heating a mixture of thiocarbohydrzide and appropriate carboxylic acids. Reaction of thiocarbohydrazide with γ-ketoesters in the presence of sodium methoxide furnished triazolopyridazine derivat...

Journal: :Antimicrobial agents and chemotherapy 1995
L J Utrup T D Moore P Actor J A Poupard

Neither amoxicillin nor clavulanic acid used alone was active at the highest level tested, i.e., 256.0 micrograms/ml, in vitro against 24 isolates of Mycobacterium fortuitum, Mycobacterium kansasii, and Mycobacterium marinum. However, the MIC of an amoxicillin-clavulanic acid combination of 2:1 was < or = 8.0/4.0 micrograms/ml for 50 percent of the isolates tested, with all isolates being inhib...

Journal: :Letters in Applied Microbiology 2005

2014
Takahiro Takazono Shigeki Nakamura Yoshifumi Imamura Taiga Miyazaki Koichi Izumikawa Hiroshi Kakeya Katsunori Yanagihara Shigeru Kohno

BACKGROUND Biological agents such as tumor necrosis factor-α inhibitors are known to cause mycobacterium infections. Here, we report a disseminated non-tuberculosis case caused by TNF-α inhibitor therapy and a probable paradoxical response to antimycobacterial therapy. CASE PRESENTATION A 68-year-old man with relapsing polychondritis was refractory to glucocorticoid therapy; adalimumab was th...

Journal: :The Journal of infectious diseases 2013
Damon P Eisen Emma S McBryde Anna Walduck

TO THE EDITOR—The report on the intrinsic antimycobacterial activity of ibupro-fen and low-dose aspirin in a novel murine tuberculosis model is fascinating

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