نتایج جستجو برای: prodynorphin

تعداد نتایج: 277  

Journal: :Pharmacological reviews 2014
Hans Jürgen Solinski Thomas Gudermann Andreas Breit

Signaling by heptahelical G protein-coupled receptors (GPCR) regulates many vital body functions. Consequently, dysfunction of GPCR signaling leads to pathologic states, and approximately 30% of all modern clinical drugs target GPCR. One decade ago, an entire new GPCR family was discovered, which was recently named MAS-related G protein-coupled receptors (MRGPR) by the HUGO Gene Nomenclature Co...

Journal: :The Journal of clinical investigation 2013
Michael Michaelides Sarah Ann R Anderson Mala Ananth Denis Smirnov Panayotis K Thanos John F Neumaier Gene-Jack Wang Nora D Volkow Yasmin L Hurd

The ability to map the functional connectivity of discrete cell types in the intact mammalian brain during behavior is crucial for advancing our understanding of brain function in normal and disease states. We combined designer receptor exclusively activated by designer drug (DREADD) technology and behavioral imaging with μPET and [18F]fluorodeoxyglucose (FDG) to generate whole-brain metabolic ...

Journal: :The international journal of neuropsychopharmacology 2013
Victor M Karpyak Stacey J Winham Ulrich W Preuss Peter Zill Julie M Cunningham Denise L Walker Kriste A Lewis Jennifer R Geske Colin L Colby Osama A Abulseoud Daniel K Hall-Flavin Larissa L Loukianova Terry D Schneekloth Mark A Frye Igor Bazov John A Heit Georgy Bakalkin David A Mrazek Joanna M Biernacka

Synthetic κ-opioid receptor (KOR) agonists induce dysphoric and pro-depressive effects and variations in the KOR (OPRK1) and prodynorphin (PDYN) genes have been shown to be associated with alcohol dependence. We genotyped 23 single nucleotide polymorphisms (SNPs) in the PDYN and OPRK1 genes in 816 alcohol-dependent subjects and investigated their association with: (1) negative craving measured ...

2012
John Moffett Linley M Fray Nicole J Kubat

BACKGROUND Pulsed radiofrequency energy (PRFE) fields are being used increasingly for the treatment of pain arising from dermal trauma. However, despite their increased use, little is known about the biological and molecular mechanism(s) responsible for PRFE-mediated analgesia. In general, current therapeutics used for analgesia target either endogenous factors involved in inflammation, or act ...

Journal: :Proceedings of the National Academy of Sciences of the United States of America 1988
M H Vilijn P J Vaysse R S Zukin J A Kessler

Expression of preproenkephalin mRNA by developing glia and neurons was examined in cultures of embryonic and neonatal rat brain. Cultured glia from specific regions of embryonic day 17 and neonatal day 1 rat brain were identified as astrocytes on the basis of both morphology and expression of immunoreactivity for glial fibrillary acidic protein. The level of preproenkephalin mRNA in cultured ne...

Journal: :The Journal of biological chemistry 2001
P B Danielson M T Hoversten M Fitzpatrick C Schreck H Akil R M Dores

The elucidation of the cDNA sequence for sturgeon proorphanin provides a unique window for interpreting the evolutionary history of the opioid/orphanin gene family. The molecular "fossil" status of this precursor can be seen in several ancestral sequence characteristics that point to its origin as a duplication of either a prodynorphin- or proenkephalin-like gene. The sturgeon proorphanin cDNA ...

Journal: :Journal of neurochemistry 2007
Jonathan Brouillette Deborah Young Matthew J During Rémi Quirion

Scopolamine-treated rats are commonly used as a psychopharmacological model of memory dysfunction and have been extensively studied to establish the effectiveness of acetylcholinesterase inhibitors in the treatment of Alzheimer's disease. Scopolamine is a muscarinic acetylcholine receptor antagonist that induces memory deficits in young subjects similar to those occurring during aging. The amne...

Journal: :Brain : a journal of neurology 2005
Thomas Carlsson Christian Winkler Corinna Burger Nicholas Muzyczka Ronald J Mandel Angela Cenci Anders Björklund Deniz Kirik

Dyskinesias are a major complication of long-term l-3,4-dihydroxyphenylalanine (L-DOPA) treatment in Parkinson's disease, and are believed to result from the intermittent and pulsatile supply of L-DOPA. Daily injections of L-DOPA can prime similar abnormal involuntary movements of the limb, orolingual and axial muscles in rats rendered parkinsonian by destruction of the nigrostriatal dopamine (...

2015
Margaret B. Allison Christa M. Patterson Michael J. Krashes Bradford B. Lowell Martin G. Myers David P. Olson

OBJECTIVE Leptin acts via its receptor (LepRb) on multiple subpopulations of LepRb neurons in the brain, each of which controls specific aspects of energy balance. Despite the importance of LepRb-containing neurons, the transcriptome and molecular identity of many LepRb subpopulations remain undefined due to the difficulty of studying the small fraction of total cells represented by LepRb neuro...

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