نتایج جستجو برای: pparδ

تعداد نتایج: 380  

2017
Katrine Qvortrup Jakob F. Jensen Mikael S. Sørensen Irene Kouskoumvekaki Rasmus K. Petersen Olivier Taboureau Karsten Kristiansen Thomas E. Nielsen

Peroxisome proliferator-activated receptor γ (PPARγ) is a well-known target for thiazolidinedione antidiabetic drugs. In this paper, we present the synthesis and biological evaluation of a series of dihydropyrano[2,3-c]pyrazole derivatives as a novel family of PPARγ partial agonists. Two analogues were found to display high affinity for PPARγ with potencies in the micro molar range. Both of the...

Journal: :Bioscience, biotechnology, and biochemistry 2013
Nobuyasu Matsuura Kanae Gamo Hiroyuki Miyachi Munekazu Iinuma Teruo Kawada Nobuyuki Takahashi Yukihiro Akao Hideki Tosa

We tested the peroxisome proliferator-activated receptor (PPAR)δ agonistic activity of a Garcinia mangostana pericarp extract to develop a treatment for the metabolic syndrome, and demonstrated γ-mangostin to be an active compound on the basis of a luciferase reporter gene assay. γ-Mangostin induced the expression of the uncoupling protein-3 (UCP-3) gene which is related to energy expenditure a...

نمودار تعداد نتایج جستجو در هر سال

با کلیک روی نمودار نتایج را به سال انتشار فیلتر کنید