نتایج جستجو برای: phthalazine

تعداد نتایج: 192  

Journal: :Cancer research 2000
J M Wood G Bold E Buchdunger R Cozens S Ferrari J Frei F Hofmann J Mestan H Mett T O'Reilly E Persohn J Rösel C Schnell D Stover A Theuer H Towbin F Wenger K Woods-Cook A Menrad G Siemeister M Schirner K H Thierauch M R Schneider J Drevs G Martiny-Baron F Totzke

PTK787/ZK 222584 (1-[4-chloroanilino]-4-[4-pyridylmethyl] phthalazine succinate) is a potent inhibitor of vascular endothelial growth factor (VEGF) receptor tyrosine kinases, active in the submicromolar range. It also inhibits other class III kinases, such as the platelet-derived growth factor (PDGF) receptor beta tyrosine kinase, c-Kit, and c-Fms, but at higher concentrations. It is not active...

Journal: :Drug metabolism and disposition: the biological fate of chemicals 2006
Lorenz M Jost Hans-Peter Gschwind Tarja Jalava Yongyu Wang Clemens Guenther Claire Souppart Antje Rottmann Karsten Denner Felix Waldmeier Gerhard Gross Eric Masson Dirk Laurent

Vatalanib (PTK787/ZK-222584) is a new oral antiangiogenic molecule that inhibits all known vascular endothelial growth factor receptors. Vatalanib is under investigation for the treatment of solid tumors. Disposition and biotransformation of vatalanib were studied in an open-label, single-center study in patients with advanced cancer. Seven patients were given a single oral (14)C-radiolabeled d...

The surface ofFe3O4 magnetic nanoparticles (MNPs) was modified by L-cysteine through condensation of COOH groups of L-cysteine and OH groups on the surface of Fe3O4. The –SH group of preparedFe3O4@Cys MNPs oxidized to –SO3H group and Fe3O4@Cys–SO3H as an environmentally friendly ...

Journal: :Physical chemistry chemical physics : PCCP 2015
Shang-Hui Ye Tian-Qing Hu Zhou Zhou Min Yang Mei-Han Quan Qun-Bo Mei Bang-Cheng Zhai Zhen-Hong Jia Wen-Yong Lai Wei Huang

Low cost and high performance white polymer light-emitting diodes (PLEDs) are very important as solid-state lighting sources. In this research three commercially available phosphors were carefully chosen, bis[2-(4,6-difluorophenyl)pyridinato-N,C(2)](picolinate)iridium(III) (FIrpic), bis[2-(2-pyridinyl-N)phenyl-C](2,4-pentanedionato-O(2),O(4))iridium(III) [Ir(ppy)2(acac)], and bis(2-phenyl-benzo...

نمودار تعداد نتایج جستجو در هر سال

با کلیک روی نمودار نتایج را به سال انتشار فیلتر کنید