نتایج جستجو برای: non glycemic benefit of sglt2 inhibitors

تعداد نتایج: 21302088  

2017
Takahiro Tosaki Hideki Kamiya Tatsuhito Himeno Yoshiro Kato Masaki Kondo Kaori Toyota Tomoyo Nishida Megumi Shiroma Kaori Tsubonaka Hitomi Asai Miho Moribe Yuki Nakaya Jiro Nakamura

Objective and Methods An SGLT2 inhibitor (ipragliflozin, dapagliflozin, luseogliflozin, tofogliflozin, or canagliflozin) was administered to 132 outpatients with type 2 diabetes mellitus with or without other antidiabetic drugs for 6 months to evaluate its efficacy, the incidence of adverse events, and its influence on the renal function. Results The patient's mean glycated hemoglobin level sig...

2017
Mehul Desai Yshai Yavin Dainius Balis Don Sun John Xie William Canovatchel Norm Rosenthal

The incidence of renal-related adverse events (AEs) with canagliflozin in patients with type 2 diabetes mellitus from a pooled population of patients in 7 active- and placebo-controlled trials (N = 5598) and in a 104-week study vs glimepiride (N = 1450) was low and similar in canagliflozin and non-canagliflozin groups. In the study vs glimepiride, canagliflozin was associated with an initial ac...

Journal: :American journal of physiology. Lung cellular and molecular physiology 2015
Ying Han Young-Eun Cho Ramon Ayon Rui Guo Katia D Youssef Minglin Pan Anzhi Dai Jason X-J Yuan Ayako Makino

Inhibitors of sodium-glucose cotransporter (SGLT)2 are a new class of oral drugs for type 2 diabetic patients that reduce plasma glucose levels by inhibiting renal glucose reabsorption. There is increasing evidence showing the beneficial effect of SGLT2 inhibitors on glucose control; however, less information is available regarding the impact of SGLT2 inhibitors on cardiovascular outcomes. The ...

2016
Simon A. Hawley Rebecca J. Ford Brennan K. Smith Graeme J. Gowans Sarah J. Mancini Ryan D. Pitt Emily A. Day Ian P. Salt Gregory R. Steinberg Grahame Hardie

Canagliflozin, dapagliflozin and empagliflozin, all recently approved for treatment of Type 2 diabetes, were derived from the natural product phlorizin. They reduce hyperglycemia by inhibiting glucose reuptake by SGLT2 in the kidney, without affecting intestinal glucose uptake by SGLT1. We now report that canagliflozin also activates AMP-activated protein kinase (AMPK), an effect also seen with...

Journal: :The Journal of pharmacology and experimental therapeutics 2012
Masayuki Suzuki Kiyofumi Honda Masanori Fukazawa Kazuharu Ozawa Hitoshi Hagita Takahiro Kawai Minako Takeda Tatsuo Yata Mio Kawai Taku Fukuzawa Takamitsu Kobayashi Tsutomu Sato Yoshiki Kawabe Sachiya Ikeda

Sodium/glucose cotransporter 2 (SGLT2) is the predominant mediator of renal glucose reabsorption and is an emerging molecular target for the treatment of diabetes. We identified a novel potent and selective SGLT2 inhibitor, tofogliflozin (CSG452), and examined its efficacy and pharmacological properties as an antidiabetic drug. Tofogliflozin competitively inhibited SGLT2 in cells overexpressing...

Journal: :Handbook of experimental pharmacology 2011
Rolf K H Kinne Francisco Castaneda

Recently, the idea has been developed to lower blood glucose blood glucose levels in diabetes by inhibiting sugar reabsorption sugar reabsorption in the kidney kidney . The main target is thereby the early proximal tubule proximal tubule where secondary active transport secondary active transport of the sugar is mediated by the sodium-D: -glucose D-glucose cotransporter SGLT2 SGLT2 . A model su...

Journal: :World Journal of Diabetes 2021

Background The efficacy of novel glucose-lowering drugs in treating non-alcoholic fatty liver disease (NAFLD) is unknown. Aim To evaluate the dipeptidyl peptidase-4 (DPP-4) inhibitors, glucagon-like peptide-1 receptor agonists (GLP-1 RAs), and sodium-glucose cotransporter 2 (SGLT2) inhibitors NAFLD to perform a comparison between these treatments. Methods Electronic databases were systematicall...

Journal: :Nature Reviews Cardiology 2017

نمودار تعداد نتایج جستجو در هر سال

با کلیک روی نمودار نتایج را به سال انتشار فیلتر کنید