نتایج جستجو برای: cyclooxygenase inhibition

تعداد نتایج: 338637  

Journal: :Circulation research 2008
Eric Arehart Jeremiah Stitham Folkert W Asselbergs Karen Douville Todd MacKenzie Kristina M Fetalvero Scott Gleim Zsolt Kasza Yamini Rao Laurie Martel Sharon Segel John Robb Aaron Kaplan Michael Simons Richard J Powell Jason H Moore Eric B Rimm Kathleen A Martin John Hwa

Recent increased adverse cardiovascular events observed with selective cyclooxygenase-2 inhibition led to the withdrawal of rofecoxib (Vioxx) and valdecoxib (Bextra), but the mechanisms underlying these atherothrombotic events remain unclear. Prostacyclin is the major end product of cyclooxygenase-2 in vascular endothelium. Using a naturally occurring mutation in the prostacyclin receptor, we r...

Journal: :Structural Chemistry 2022

Inhibition of microsomal prostaglandin E2 synthase-1 (mPGES-1) is promising for designing novel nonsteroidal anti-inflammatory drugs, as they lack side-effects associated with inhibition cyclooxygenase enzymes. Azole compounds are nitrogen-containing heterocycles and have a wide use in medicine considered medicinal chemistry. Various computer-aided drug design strategies incorporated this study...

Journal: :Journal of applied physiology 2005
Jennifer M Lockwood Mollie P Pricher Brad W Wilkins Lacy A Holowatz John R Halliwill

In normally active individuals, postexercise hypotension after a single bout of aerobic exercise occurs due to an unexplained peripheral vasodilation. Prostaglandin production has been suggested to contribute to the increases in blood flow during and after exercise; however, its potential contribution to postexercise hypotension has not been assessed. The purpose of this study was to determine ...

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